SCHEMBL18600155

SCHEMBL18600155

C#CCN(Cc1ccc(F)cc1)c1ccc(NC)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 4/20 0.53
KCNQ4 P56696 4/20 0.52
KCNQ5 Q9NR82 3/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C8 P10632 1/20 0.51
CYP2B6 P20813 1/20 0.51
KCNQ2 O43526 1/20 0.49
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
TYMS P04818 2/20 0.36
DHFR P00374 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15997126 0.87 KCNQ4 (0.53) PYCR1KCNQ4KCNQ5CYP1A2CYP2C8
SCHEMBL30494445 0.82 KCNQ4 (0.60) PYCR1KCNQ4KCNQ5CYP1A2CYP2C8
SCHEMBL15996890 0.82 CYP1A2 (0.72) PYCR1KCNQ4KCNQ5CYP1A2CYP2C8
SCHEMBL18575368 0.82 KCNQ4 (0.59) PYCR1KCNQ4KCNQ5CYP1A2CYP2C8
SCHEMBL20159076 0.81 KCNQ4 (0.56) PYCR1KCNQ4KCNQ5CYP1A2CYP2C8
SCHEMBL15996915 0.81 PYCR1 (0.53) PYCR1KCNQ4KCNQ5CYP1A2CYP2C8
SCHEMBL23969465 0.80 CYP1A2 (0.49) PYCR1KCNQ4KCNQ5CYP1A2CYP2C8
SCHEMBL18600341 0.80 KCNQ4 (0.55) PYCR1KCNQ4KCNQ5CYP1A2CYP2C8
SCHEMBL18600345 0.79 CYP1A2 (0.59) PYCR1KCNQ4KCNQ5CYP1A2CYP2C8
SCHEMBL18575369 0.79 ALDH1A1 (0.61) PYCR1KCNQ4KCNQ5CYP1A2CYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3138833-A1 NOVEL KCNQ POTASSIUM CHANNEL AGONIST, AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2017-03-08 EP disclosed