SCHEMBL18600372

SCHEMBL18600372

C#CCNc1cc(C)c(NC(=O)OC)c(C)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.48
CYP2C8 P10632 1/20 0.48
CYP2B6 P20813 1/20 0.48
NLRP3 Q96P20 2/20 0.40
LCK P06239 1/20 0.37
CA12 O43570 2/20 0.37
CA9 Q16790 2/20 0.37
CA4 P22748 1/20 0.37
HPGD P15428 2/20 0.37
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
LMNA P02545 1/20 0.35
HSD17B10 Q99714 2/20 0.35
PTPRB P23467 1/20 0.35
TSHR P16473 1/20 0.35
MAPT P10636 2/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
KDM4E B2RXH2 1/20 0.34
USP2 O75604 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28098568 0.77 SMN1; SMN2 (0.56) CA12CA9HPGDALDH1A1SMN1; SMN2
SCHEMBL2089479 0.74 NLRP3 (0.59) NLRP3LCKHPGDALDH1A1LMNA
SCHEMBL18600165 0.73 CYP1A2 (0.55) CYP1A2CYP2C8CYP2B6ALDH1A1SMN1; SMN2
SCHEMBL18600164 0.71 HPGD (0.44) CYP1A2CYP2C8CYP2B6NLRP3LCK
SCHEMBL31059176 0.71 MAPT (0.54) CYP1A2CYP2C8CYP2B6NLRP3LCK
SCHEMBL16234657 0.71 MAPT (0.44) CYP1A2CYP2C8CYP2B6CA12CA9
SCHEMBL5184928 0.70 CYP1A2 (0.44) CYP1A2CYP2C8CYP2B6HPGDALDH1A1
SCHEMBL31738102 0.67 KDM4E (0.37) CYP1A2CA12CA9HPGDALDH1A1
SCHEMBL2096567 0.66 NLRP3 (0.59) CYP1A2NLRP3ALDH1A1LMNATSHR
SCHEMBL11510151 0.66 RAF1 (0.45) CYP1A2CYP2C8CYP2B6NLRP3LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3138833-A1 NOVEL KCNQ POTASSIUM CHANNEL AGONIST, AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2017-03-08 EP disclosed