SCHEMBL18601657

SCHEMBL18601657

[CH2]CCNCc1ccc(OCCCCCc2ccccc2)c(-c2ncco2)c1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BCHE P06276 6/20 0.40
ROCK1 Q13464 2/20 0.39
ROCK2 O75116 1/20 0.39
KCNH2 Q12809 1/20 0.39
SIGMAR1 Q99720 3/20 0.39
SLC2A1 P11166 1/20 0.38
S1PR1 P21453 3/20 0.37
S1PR3 Q99500 1/20 0.37
S1PR5 Q9H228 1/20 0.37
FAAH O00519 1/20 0.36
CES1 P23141 1/20 0.36
NCEH1 Q6PIU2 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2385767 0.85 S1PR1 (0.51) S1PR1S1PR3S1PR5
SCHEMBL18601658 0.85 SIGMAR1 (0.41) BCHEROCK1ROCK2KCNH2SIGMAR1
SCHEMBL15042521 0.85 S1PR1 (0.39) BCHESIGMAR1SLC2A1S1PR1S1PR3
SCHEMBL18601656 0.81 SIGMAR1 (0.40) BCHEROCK1ROCK2KCNH2SIGMAR1
SCHEMBL18601666 0.80 SLC6A9 (0.39) BCHEROCK1ROCK2KCNH2SIGMAR1
SCHEMBL18601662 0.78 SIGMAR1 (0.40) BCHESIGMAR1SLC2A1S1PR1S1PR3
SCHEMBL18601653 0.77 HTR1A (0.45) BCHESIGMAR1SLC2A1S1PR1S1PR3
SCHEMBL18601654 0.77 HTR1A (0.45) BCHESIGMAR1SLC2A1
SCHEMBL1977951 0.74 S1PR5 (0.49) S1PR1S1PR3S1PR5
SCHEMBL15042627 0.72 BCHE (0.39) BCHEROCK1SIGMAR1S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2504323-B1 NOVEL COMPOUNDS AS RECEPTOR MODULATORS WITH THERAPEUTIC UTILITY ALLERGAN INC (US) 2017-03-15 EP claimed