SCHEMBL18601663

SCHEMBL18601663

[CH2]CCNCc1ccc(OCCCCCc2ccccc2)c(-c2cccs2)n1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 4/20 0.38
SIGMAR1 Q99720 3/20 0.36
DAGLA Q9Y4D2 1/20 0.36
FAAH O00519 1/20 0.36
CES1 P23141 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.34
HDAC1 Q13547 1/20 0.34
BCHE P06276 1/20 0.33
NTRK3 Q16288 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1979185 0.85 S1PR3 (0.49)
SCHEMBL15042602 0.85 HDAC1 (0.36) NR1H4SIGMAR1DAGLAFAAHCES1
SCHEMBL18601662 0.80 SIGMAR1 (0.40) SIGMAR1BCHE
SCHEMBL12760665 0.80 PLAU (0.38) NR1H4SIGMAR1SMN1; SMN2BCHE
SCHEMBL15022995 0.71 C5AR1 (0.40) SIGMAR1FAAHCES1BCHE
SCHEMBL18601666 0.71 SLC6A9 (0.39) SIGMAR1CES1BCHE
SCHEMBL15023492 0.70 SIGMAR1 (0.44) SIGMAR1BCHE
SCHEMBL1979687 0.68 SIGMAR1 (0.41) SIGMAR1BCHE
SCHEMBL18601655 0.68 C5AR1 (0.39) SIGMAR1SMN1; SMN2BCHE
SCHEMBL18601659 0.67 S1PR2 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2504323-B1 NOVEL COMPOUNDS AS RECEPTOR MODULATORS WITH THERAPEUTIC UTILITY ALLERGAN INC (US) 2017-03-15 EP claimed