SCHEMBL18609481

SCHEMBL18609481

c1ccc(-n2cnc3ccc(-c4cn[nH]c4)cc32)cc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.53
ALDH1A1 P00352 1/20 0.53
HPGD P15428 1/20 0.53
MAPK1 P28482 1/20 0.53
MAPK10 P53779 1/20 0.53
NCOA1 Q15788 1/20 0.53
NCOA3 Q9Y6Q9 1/20 0.53
ATM Q13315 3/20 0.53
FGFR1 P11362 4/20 0.50
GRK2 P25098 2/20 0.50
GRK1 Q15835 2/20 0.50
GRK5 P34947 1/20 0.50
KDR P35968 1/20 0.49
SRC P12931 2/20 0.48
AKT1 P31749 1/20 0.46
AKT2 P31751 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3847802 0.86 ATM (0.45) ATMGRK2GRK1GRK5
SCHEMBL18609350 0.85 FGFR1 (0.56) HPGDATMFGFR1GRK2GRK1
SCHEMBL18609278 0.84 GABRP (0.43) ATMGRK2GRK1GRK5
SCHEMBL16291053 0.82 HTT (0.62) HTTALDH1A1HPGDMAPK1MAPK10
SCHEMBL18609277 0.82 FGFR1 (0.47) ATMFGFR1GRK2GRK1GRK5
SCHEMBL18609354 0.80 FGFR1 (0.59) ATMFGFR1SRC
SCHEMBL12822377 0.80 GP6 (0.41) ALDH1A1ATMGRK2GRK1GRK5
SCHEMBL22070428 0.80 MAP3K8 (0.41) HTTALDH1A1HPGDMAPK1MAPK10
SCHEMBL18584433 0.78 HCAR1 (0.52) ATMFGFR1GRK2GRK1GRK5
SCHEMBL19228785 0.77 HTT (0.56) HTTALDH1A1HPGDMAPK1MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017040993-A1 SMALL MOLECULE INHIBITORS OF DYRK1A AND USES THEREOF THE ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2017-03-09 WO disclosed