SCHEMBL18616895

SCHEMBL18616895

c1cc(Nc2ccc(-c3nc4cc(Nc5ccncc5)ccc4[nH]3)cc2)ccn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.51
KDM4E B2RXH2 4/20 0.51
PKN1 Q16512 4/20 0.51
PKN2 Q16513 4/20 0.51
HPGD P15428 3/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
HSD17B10 Q99714 1/20 0.51
RHEB Q15382 1/20 0.51
GAA P10253 1/20 0.48
HPSE Q9Y251 3/20 0.47
NPC1 O15118 4/20 0.47
RAB9A P51151 3/20 0.47
GUSB P08236 1/20 0.45
KMT2A Q03164 2/20 0.44
PKM P14618 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL18586196 0.98 ALDH1A1 (0.50) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL24011225 0.93 RAD52 (0.53) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL23999512 0.89 MEN1 (0.54) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL30440947 0.85 KDM4E (0.73) ALDH1A1KDM4EPKN1PKN2HPGD
Hydrochloric Acid SCHEMBL18585474 0.85 MAPKAPK2 (0.49)
SCHEMBL18585635 0.84 ROCK2 (0.54) ALDH1A1KDM4EHPGDCYP1A2CYP3A4
SCHEMBL18617611 0.84 NPC1 (0.43) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL18617883 0.83 KDM4E (0.38) ALDH1A1KDM4EPKN1PKN2HPGD
Hydrochloric Acid SCHEMBL18585863 0.83 NPC1 (0.42) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL23999511 0.81 KDR (0.63) ALDH1A1KDM4EHPGDCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017039318-A1 BENZIMIDAZOLE DERIVATIVES FOR DNA METHYLATION INHIBITORS KAINOS MEDICINE, INC. (KR) 2017-03-09 WO disclosed