SCHEMBL186281

SCHEMBL186281

Cc1cc(Nc2ccc(F)cc2C(F)(F)F)cnc1CNC(=O)[C@]1(NC(=O)Oc2cncnc2)CCOC1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 3/20 0.36
CNR2 P34972 2/20 0.31
FAAH O00519 2/20 0.31
TRPV1 Q8NER1 1/20 0.31
DHODH Q02127 1/20 0.30
NTRK1 P04629 1/20 0.30
P2RX7 Q99572 2/20 0.30
MKNK2 Q9HBH9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL185516 0.94 OPRL1 (0.36) OPRL1CNR2FAAHTRPV1DHODH
SCHEMBL14856439 0.93 FAAH (0.33) OPRL1CNR2FAAHTRPV1DHODH
SCHEMBL186543 0.92 OPRL1 (0.34) OPRL1CNR2FAAHTRPV1P2RX7
SCHEMBL2805695 0.91 OPRL1 (0.37) OPRL1CNR2DHODH
SCHEMBL185881 0.88 OPRL1 (0.37) OPRL1CNR2FAAHTRPV1P2RX7
SCHEMBL185388 0.88 OPRL1 (0.36) OPRL1CNR2FAAHTRPV1NTRK1
SCHEMBL186992 0.87 CNR2 (0.33) CNR2FAAHTRPV1P2RX7
SCHEMBL186076 0.87 CNR2 (0.37) CNR2FAAHTRPV1DHODHP2RX7
SCHEMBL14856590 0.86 FAAH (0.35) OPRL1CNR2FAAHTRPV1DHODH
SCHEMBL186188 0.86 CNR2 (0.35) CNR2FAAHTRPV1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-01-04 EP disclosed
WO-2010097372-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed