SCHEMBL18638656

SCHEMBL18638656

CC(C)(O)CN1CNc2cc(-c3ccccc3Cl)ccc21

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PGR P06401 3/20 0.34
PDK2 Q15119 2/20 0.34
PAK1 Q13153 2/20 0.34
SCN9A Q15858 1/20 0.33
TNKS2 Q9H2K2 1/20 0.33
CNR2 P34972 1/20 0.33
MCHR1 Q99705 1/20 0.33
PDK1 Q15118 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
USP30 Q70CQ3 1/20 0.33
GRM2 Q14416 1/20 0.33
TRPA1 O75762 1/20 0.33
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
TYK2 P29597 1/20 0.32
JAK3 P52333 1/20 0.32
GSK3B P49841 1/20 0.32
MAPK14 Q16539 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18638458 0.91 PGR (0.36) PGRPDK2PAK1SCN9ATNKS2
SCHEMBL18638345 0.89 RORC (0.37) SCN9A
SCHEMBL18638341 0.87 MARS1 (0.38) PDK2PDK1PDK3PDK4
SCHEMBL18638652 0.83 GRM2 (0.36) PDK2GRM2
SCHEMBL18638655 0.82 PGR (0.41) PGRCNR2GRM2
SCHEMBL18638344 0.81 ABL1 (0.32)
SCHEMBL18638339 0.81 FASN (0.34) SCN9AGRM2
SCHEMBL18638640 0.80 RORC (0.37) SCN9A
SCHEMBL18638639 0.78 AHR (0.36) PDK2PDK1PDK3PDK4MAPK14
SCHEMBL18638664 0.76 APP (0.42) GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017043636-A1 NOVEL BENZIMIDAZOLE COMPOUND AND PHARMACEUTICAL USE OF SAME 大日本住友製薬株式会社 2017-03-16 WO disclosed