SCHEMBL18639909

SCHEMBL18639909

CCN1CCC(COc2ccc3c(N)n[nH]c3c2)CC1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.44
MAOB P27338 3/20 0.41
MAOA P21397 2/20 0.41
SIGMAR1 Q99720 2/20 0.41
LRRK2 Q5S007 1/20 0.40
PARP15 Q460N3 1/20 0.40
PARP10 Q53GL7 1/20 0.40
ACHE P22303 2/20 0.39
ALB P02768 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18639981 0.88 MAOA (0.50) CHEK1MAOBMAOAPARP15PARP10
SCHEMBL18639866 0.86 PARP15 (0.51) MAOBMAOAPARP15PARP10
SCHEMBL18639974 0.85 CHEK1 (0.45) CHEK1MAOBMAOAPARP15PARP10
SCHEMBL18640109 0.84 PARP10 (0.53) MAOBMAOAPARP15PARP10
SCHEMBL18640024 0.83 CYP4F2 (0.53) LRRK2
SCHEMBL18640136 0.83 PARP10 (0.54) MAOBMAOAPARP15PARP10
SCHEMBL18639947 0.82 F10 (0.54) MAOBMAOAACHE
SCHEMBL18639846 0.82 CYP4F2 (0.41) PARP15PARP10
SCHEMBL18639875 0.82 DRD2 (0.43)
SCHEMBL18639956 0.82 SLC6A2 (0.53) MAOBMAOAPARP15PARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017045751-A1 COMPOUNDS AS ASIC INHIBITORS AND USES THEREOF MERCK PATENT GMBH (DE) 2017-03-23 WO disclosed
WO-2017045751-A1 COMPOUNDS AS ASIC INHIBITORS AND USES THEREOF MERCK PATENT GMBH (DE) 2017-03-23 WO disclosed