SCHEMBL18644682

SCHEMBL18644682

C/C=C(/Br)c1sc(C(C)=O)nc1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.38
SMN1; SMN2 Q16637 6/20 0.38
RAB9A P51151 6/20 0.37
NPC1 O15118 6/20 0.37
MAPT P10636 4/20 0.37
RXFP1 Q9HBX9 2/20 0.36
CYP1A2 P05177 1/20 0.36
GAA P10253 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 2/20 0.35
TSHR P16473 2/20 0.35
KMT2A Q03164 5/20 0.34
KDM4E B2RXH2 3/20 0.34
MEN1 O00255 3/20 0.34
PKM P14618 1/20 0.33
POLB P06746 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18644683 0.83 ALDH1A1 (0.42) ALDH1A1SMN1; SMN2RAB9ANPC1MAPT
SCHEMBL18644693 0.83 ALDH1A1 (0.40) ALDH1A1RAB9ANPC1MAPTHPGD
SCHEMBL13165457 0.82 RXFP1 (0.49) ALDH1A1SMN1; SMN2RAB9ANPC1MAPT
SCHEMBL27829742 0.79 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2RAB9ANPC1MAPT
SCHEMBL27848208 0.71 ALDH1A1 (0.60) ALDH1A1RAB9ANPC1MAPTCYP1A2
SCHEMBL569821 0.71 NOS1 (0.41) ALDH1A1SMN1; SMN2RAB9ANPC1MAPT
SCHEMBL18355569 0.70 SMN1; SMN2 (0.37) ALDH1A1SMN1; SMN2RAB9ANPC1MAPT
SCHEMBL3000943 0.69 SMN1; SMN2 (0.45) ALDH1A1SMN1; SMN2RAB9ANPC1MAPT
SCHEMBL18644689 0.69 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2RAB9ANPC1MAPT
SCHEMBL3655946 0.66 ALDH1A1 (0.61) ALDH1A1SMN1; SMN2RAB9ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9617279-B1 Imidazooxadiazole compounds BRISTOL-MYERS SQUIBB COMPANY (US) 2017-04-11 US disclosed
US-9598419-B1 Imidazotriazine and imidazodiazine compounds UNIVERSITE DE MONTREAL (CA) 2017-03-21 US disclosed