SCHEMBL18654355

SCHEMBL18654355

NNC(=O)C(=O)Nc1cccc(N2CCC2)n1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 11/20 0.46
CNR2 P34972 1/20 0.46
HSD11B1 P28845 2/20 0.41
CDK5 Q00535 1/20 0.41
CDK5R1 Q15078 1/20 0.41
KIF18A Q8NI77 2/20 0.40
OGA O60502 1/20 0.39
FAAH O00519 1/20 0.38
AOC3 Q16853 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
TYK2 P29597 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14879935 0.84 CNR1 (0.49) CNR1CNR2HSD11B1CDK5CDK5R1
SCHEMBL28879200 0.82 CNR1 (0.49) CNR1CNR2HSD11B1CDK5CDK5R1
SCHEMBL29805447 0.78 CNR1 (0.46) CNR1CNR2HSD11B1CDK5CDK5R1
SCHEMBL23451255 0.78 ADORA2A (0.55) CNR1CNR2HSD11B1CDK5CDK5R1
SCHEMBL18654609 0.75 CNR1 (0.40) CNR1CNR2HSD11B1CDK5CDK5R1
SCHEMBL2566436 0.72 HSD11B1 (0.64) CNR1HSD11B1AOC3
SCHEMBL22146027 0.72 NUDT1 (0.47) CNR1CNR2HSD11B1TYK2
SCHEMBL2950708 0.70 CNR1 (0.45) CNR1CNR2HSD11B1CDK5CDK5R1
SCHEMBL23599390 0.69 NPC1 (0.49) CNR1CNR2AOC3
SCHEMBL20688213 0.68 CNR1 (0.44) CNR1CNR2HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2768509-B1 SUBSTITUTED BICYCLIC AZA-HETEROCYCLES AND ANALOGUES AS SIRTUIN MODULATORS GLAXOSMITHKLINE LLC (US) 2017-03-22 EP disclosed