SCHEMBL18655372

SCHEMBL18655372

COc1cc(C2=C(c3cn(CCCNC(=O)C(N)CO)c4ccccc34)C(=O)NC2=O)cc(O)c1OC

nearest known ligand 0.80

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 11/20 0.80
KDR P35968 11/20 0.66
FLT3 P36888 8/20 0.66
QPCT Q16769 1/20 0.49
CAMK2D Q13557 3/20 0.47
PLK4 O00444 1/20 0.46
AURKA O14965 1/20 0.46
NUAK1 O60285 1/20 0.46
PDGFRB P09619 1/20 0.46
FLT4 P35916 1/20 0.46
TEK Q02763 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9954914 0.95 GSK3B (0.87) GSK3BKDRFLT3QPCTCAMK2D
SCHEMBL10069744 0.89 GSK3B (1.00) GSK3BKDRFLT3QPCTCAMK2D
SCHEMBL18655375 0.88 GSK3B (0.79) GSK3BKDRFLT3QPCTCAMK2D
SCHEMBL18655336 0.84 GSK3B (0.86) GSK3BKDRFLT3QPCTCAMK2D
SCHEMBL18655373 0.83 GSK3B (0.91) GSK3BKDRFLT3QPCTCAMK2D
SCHEMBL8540158 0.82 PIM1 (0.65) GSK3BCAMK2D
SCHEMBL10070111 0.82 GSK3B (0.68) GSK3BKDRFLT3QPCTCAMK2D
SCHEMBL18628480 0.82 GSK3B (0.68) GSK3BKDRFLT3QPCTCAMK2D
SCHEMBL18655377 0.81 GSK3B (0.91) GSK3BKDRFLT3QPCTPLK4
SCHEMBL18655354 0.81 GSK3B (0.61) GSK3BKDRFLT3QPCTCAMK2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655359-B1 CONJUGATED 3-(INDOLYL)- AND 3-(AZAINDOLYL)-4-ARYLMALEIMIDE COMPOUNDS AND THEIR USE IN TUMOR TREATMENT Johannes-Gutenberg-Universität Mainz (DE) 2017-03-22 EP disclosed