SCHEMBL18667192

SCHEMBL18667192

CCc1ncc(CNC(=O)c2ccc3c(c2)NC(=O)c2ccccc2O3)s1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 4/20 0.42
DRD2 P14416 1/20 0.40
TAOK1 Q7L7X3 1/20 0.39
ABL1 P00519 2/20 0.38
RAB9A P51151 1/20 0.37
KMT2A Q03164 3/20 0.37
ALDH1A1 P00352 2/20 0.37
POLB P06746 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MEN1 O00255 2/20 0.37
HPGD P15428 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
SLC8A1 P32418 1/20 0.36
LMNA P02545 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23018621 0.90 ALOX5 (0.41) ALOX5RAB9AALDH1A1SLC8A1LMNA
SCHEMBL18667069 0.89 ALOX5 (0.43) ALOX5DRD2TAOK1ABL1RAB9A
SCHEMBL18667324 0.88 ALOX5 (0.44) ALOX5DRD2TAOK1ABL1RAB9A
SCHEMBL30271085 0.88 ALOX5 (0.44) ALOX5DRD2TAOK1ABL1RAB9A
SCHEMBL18667886 0.87 ALOX5 (0.39) ALOX5DRD2TAOK1ABL1RAB9A
SCHEMBL30271101 0.87 ALOX5 (0.39) ALOX5DRD2TAOK1ABL1RAB9A
SCHEMBL18667193 0.86 ALOX5 (0.41) ALOX5DRD2TAOK1ABL1RAB9A
SCHEMBL30271136 0.86 DRD2 (0.51) ALOX5DRD2ABL1RAB9AKMT2A
SCHEMBL18667362 0.86 DRD2 (0.51) ALOX5DRD2ABL1RAB9AKMT2A
SCHEMBL18667545 0.85 ALOX5 (0.42) ALOX5DRD2TAOK1ABL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240025890-A1 HEPATITIS B CORE PROTEIN MODULATORS ASSEMBLY BIOSCIENCES INC (US) 2024-01-25 US disclosed
US-20240025890-A1 HEPATITIS B CORE PROTEIN MODULATORS ASSEMBLY BIOSCIENCES INC (US) 2024-01-25 US disclosed
US-11814376-B2 Hepatitis b core protein modulators ASSEMBLY BIOSCIENCES, INC. (US) 2023-11-14 US disclosed
US-11814376-B2 Hepatitis b core protein modulators ASSEMBLY BIOSCIENCES, INC. (US) 2023-11-14 US disclosed
US-20230044112-A1 HEPATITIS B CORE PROTEIN MODULATORS ASSEMBLY BIOSCIENCES, INC. (US) 2023-02-09 US disclosed
US-10968211-B2 Hepatitis B core protein modulators ASSEMBLY BIOSCIENCES, INC. (US) 2021-04-06 US disclosed
EP-3782626-A1 HEPATITIS B CORE PROTEIN MODULATORS Assembly Biosciences, Inc. (US) 2021-02-24 EP disclosed
US-20200131168-A1 HEPATITIS B CORE PROTEIN MODULATORS INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION 2020-04-30 US disclosed
US-10377748-B2 Hepatitis B core protein modulators ASSEMBLY BIOSCIENCES, INC. (US) 2019-08-13 US disclosed
WO-2017048950-A1 HEPATITIS B CORE PROTEIN MODULATORS ASSEMBLY BIOSCIENCES, INC. (US) 2017-03-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240025890-A1 HEPATITIS B CORE PROTEIN MODULATORS HAVCR2, FABP1, MAVS ALOX5 4186/4885DRD2 4229/4885TAOK1 3842/4885
US-20230044112-A1 HEPATITIS B CORE PROTEIN MODULATORS HAVCR2, FABP1, MAVS ALOX5 4186/4885DRD2 4229/4885TAOK1 3842/4885
US-10377748-B2 Hepatitis B core protein modulators HAVCR2, FABP1, MAVS ALOX5 4186/4885DRD2 4229/4885TAOK1 3842/4885
US-10968211-B2 Hepatitis B core protein modulators HAVCR2, FABP1, MAVS ALOX5 4186/4885DRD2 4229/4885TAOK1 3842/4885
US-11814376-B2 Hepatitis b core protein modulators HAVCR2, FABP1, MAVS ALOX5 4186/4885DRD2 4229/4885TAOK1 3842/4885
US-20200131168-A1 HEPATITIS B CORE PROTEIN MODULATORS HAVCR2, FABP1, MAVS ALOX5 4186/4885DRD2 4229/4885TAOK1 3842/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.