SCHEMBL18699459

SCHEMBL18699459

CCCSc1cccc(N2CCN(Cc3ccccc3)CC2)c1CC=O

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 8/20 0.46
DRD2 P14416 6/20 0.46
DRD3 P35462 6/20 0.46
MAPT P10636 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
ATM Q13315 1/20 0.40
SIGMAR1 Q99720 1/20 0.39
HTR6 P50406 1/20 0.39
HTR7 P34969 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18699453 0.84 DRD4 (0.47) DRD4DRD2DRD3MAPTNPSR1
SCHEMBL18699520 0.83 DRD4 (0.46) DRD4DRD2DRD3MAPTNPSR1
SCHEMBL18699539 0.82 DRD4 (0.51) DRD4DRD2DRD3MAPTNPSR1
SCHEMBL18699458 0.81 HTR1A (0.44) DRD4DRD2DRD3
SCHEMBL12000243 0.70 DRD4 (0.64) DRD4DRD2DRD3MAPTNPSR1
SCHEMBL18699541 0.70 DRD2 (0.48) DRD4DRD2DRD3MAPTNPSR1
SCHEMBL2597773 0.69 DRD4 (0.72) DRD4DRD2DRD3MAPTL3MBTL1
SCHEMBL418557 0.68 DRD4 (0.57) DRD4DRD2DRD3MAPTNPSR1
SCHEMBL14132945 0.67 DRD4 (0.59) DRD4DRD2DRD3MAPTNPSR1
SCHEMBL7426690 0.66 DRD4 (0.68) DRD4DRD2DRD3MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3150591-A1 PROCESS AND INTERMEDIATES FOR THE PREPARATION OF BENZO[B]THIOPHENE COMPOUNDS Crystal Pharma S.A.U (ES) 2017-04-05 EP disclosed