SCHEMBL18708221

SCHEMBL18708221

COc1cnc(C(C)=O)cc1OCC1CC1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPC6 Q9Y210 5/20 0.49
CNR2 P34972 10/20 0.45
PDE4B Q07343 5/20 0.44
PDE4A P27815 2/20 0.44
PDE4C Q08493 2/20 0.44
PDE4D Q08499 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL88281 0.88 TRPC6 (0.49) TRPC6CNR2PDE4BPDE4APDE4C
SCHEMBL71158 0.87 TRPC6 (0.48) TRPC6CNR2PDE4BPDE4APDE4C
SCHEMBL3633786 0.87 TRPC6 (0.54) TRPC6CNR2PDE4BPDE4APDE4C
SCHEMBL21045798 0.82 TRPC6 (0.55) TRPC6CNR2
Potassium Ion SCHEMBL15757775 0.81 TRPC6 (0.44) TRPC6CNR2PDE4BPDE4APDE4C
SCHEMBL30439691 0.81 TRPC6 (0.54) TRPC6CNR2
SCHEMBL21045633 0.81 TRPC6 (0.54) TRPC6CNR2
SCHEMBL15757242 0.79 PDE4B (0.41) TRPC6PDE4BPDE4APDE4CPDE4D
SCHEMBL26445599 0.78 CNR2 (0.53) CNR2
SCHEMBL72985 0.78 PDE4D (0.59) CNR2PDE4BPDE4APDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9611250-B2 Process for preparing 4-(cyclopropylmethoxy)-N-(3,5-dichloro-1-oxido-4-pyridyl)-5-methoxypyridine-2-carboxamide SANOFI (FR) 2017-04-04 US disclosed