SCHEMBL18740554

SCHEMBL18740554

O=C(N[C@@H](Cc1ccccc1)[C@H](O)CNCc1ccccc1)c1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 14/20 0.67
SLC6A11 P48066 1/20 0.67
BCHE P06276 6/20 0.60
BACE2 Q9Y5Z0 3/20 0.54
CTSD P07339 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7310941 0.93 BACE1 (0.56) BACE1SLC6A11BCHE
SCHEMBL7610032 0.87 BACE1 (0.71) BACE1SLC6A11BCHE
SCHEMBL7610027 0.87 BACE1 (0.71) BACE1SLC6A11BCHE
SCHEMBL8577646 0.86 NPC1 (0.53) BACE1SLC6A11BACE2CTSD
SCHEMBL5400472 0.85 BACE1 (0.74) BACE1BCHEBACE2CTSD
SCHEMBL5380143 0.85 BACE1 (0.77) BACE1BCHECTSD
Hydrochloric Acid SCHEMBL5382955 0.84 BACE1 (0.75) BACE1BCHECTSD
SCHEMBL8729415 0.83 BACE1 (0.67) BACE1SLC6A11BCHE
SCHEMBL6809872 0.82 CTRB1 (0.55)
SCHEMBL6814426 0.82 CTRB1 (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017066742-A1 BACE-2 INHIBITORY COMPOUNDS AND RELATED METHODS OF USE JORTAN PHARMACEUTICALS INC. (US) 2017-04-20 WO claimed
WO-2017066742-A1 BACE-2 INHIBITORY COMPOUNDS AND RELATED METHODS OF USE JORTAN PHARMACEUTICALS INC. (US) 2017-04-20 WO disclosed