SCHEMBL18754242

SCHEMBL18754242

CNC(=O)c1c(NC)cc(C)nc1C

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.38
MAPT P10636 1/20 0.35
BAZ2B Q9UIF8 1/20 0.35
GAA P10253 2/20 0.35
ALDH1A1 P00352 3/20 0.34
HPGD P15428 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
PKM P14618 2/20 0.34
LMNA P02545 1/20 0.34
RAB9A P51151 1/20 0.34
SPR P35270 1/20 0.34
MAPK1 P28482 2/20 0.33
POLB P06746 1/20 0.33
NOS3 P29474 1/20 0.33
NOS2 P35228 1/20 0.33
HSP90AB1 P08238 1/20 0.33
MEN1 O00255 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL900397 0.79 KMT2A (0.41) SMN1; SMN2MAPTALDH1A1LMNARAB9A
SCHEMBL12341497 0.70 NOS3 (0.41) MAPTGAAALDH1A1PKMMAPK1
SCHEMBL353805 0.70 PDK2 (0.43) SMN1; SMN2MAPTBAZ2BGAAALDH1A1
SCHEMBL8568255 0.69 HDAC8 (0.45) SMN1; SMN2MAPTBAZ2BALDH1A1HPGD
SCHEMBL899803 0.68 NCF1 (0.46) HPGDNPSR1
SCHEMBL26906303 0.68 MEN1 (0.46) SMN1; SMN2BAZ2BALDH1A1MAPK1POLB
SCHEMBL29827115 0.68 MEN1 (0.46) SMN1; SMN2BAZ2BALDH1A1MAPK1POLB
SCHEMBL23889492 0.67 NOS3 (0.39) SMN1; SMN2MAPTGAAALDH1A1NOS3
SCHEMBL30632136 0.67 ALDH1A1 (0.47) SMN1; SMN2GAAALDH1A1HPGDLMNA
SCHEMBL361910 0.66 POLB (0.43) MAPTGAAALDH1A1HPGDSPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3036235-B1 NEW BIS-AMIDO PYRIDINES BOEHRINGER INGELHEIM INT (DE) 2017-04-19 EP disclosed
EP-3036228-B1 NEW 6-ALKYNYL PYRIDINE COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2017-04-19 EP disclosed