SCHEMBL18763340

SCHEMBL18763340

Oc1ccc(C2CCN(Cl)CC2)cc1

nearest known ligand 0.61

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 12/20 0.61
ESR1 P03372 2/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10265387 0.81 DRD2 (0.59)
SCHEMBL28880095 0.81 ESR2 (0.63) ESR2ESR1CYP3A4CYP2C9
SCHEMBL1865798 0.79 ESR2 (0.81) ESR2ESR1CYP3A4CYP2C9
SCHEMBL1986271 0.79 ESR2 (0.81) ESR2ESR1CYP3A4CYP2C9
SCHEMBL3809909 0.79 ESR2 (0.81) ESR2ESR1CYP3A4CYP2C9
SCHEMBL3811445 0.79 ESR2 (0.81) ESR2ESR1CYP3A4CYP2C9
SCHEMBL12686989 0.79 SLC18A3 (0.53) ESR2
SCHEMBL13783635 0.79 QDPR (0.65) ESR2ESR1CYP3A4CYP2C9
SCHEMBL18255078 0.79 DRD2 (0.47)
SCHEMBL11062207 0.78 SLC18A3 (0.55) CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017066368-A1 SELECTIVE NR2B ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2017-04-20 WO disclosed