SCHEMBL1878409

SCHEMBL1878409

CC(C)(C)CN(CCC#N)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.42
MLYCD O95822 2/20 0.38
ALDH1A1 P00352 8/20 0.38
NPC1 O15118 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MAPT P10636 1/20 0.36
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.34
AR P10275 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
GAA P10253 2/20 0.33
HPGD P15428 1/20 0.33
CASP1 P29466 1/20 0.33
LIMK1 P53667 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15519635 0.83 MLYCD (0.40) POLBMLYCDALDH1A1NPC1L3MBTL1
SCHEMBL4444128 0.81 POLB (0.46) POLBMLYCDALDH1A1NPC1L3MBTL1
SCHEMBL5933411 0.78 MLYCD (0.47) POLBMLYCDALDH1A1NPC1L3MBTL1
SCHEMBL4720974 0.76 TSHR (0.33) ALDH1A1TSHRCYP2D6CYP2C19
SCHEMBL1132975 0.75 CA12 (0.31) ALDH1A1MAPT
SCHEMBL559019 0.74 PIN1 (0.33)
SCHEMBL657409 0.74 KDM4E (0.31)
SCHEMBL3706142 0.72 ALDH1A1 (0.38) POLBMLYCDALDH1A1NPC1L3MBTL1
Hydrochloric Acid SCHEMBL1026856 0.72 KDM4E (0.34)
SCHEMBL4062047 0.72 NTRK2 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2496557-A1 TETRAHYDROQUINOLINE DERIVATIVES AND THEIR PHARMACEUTICAL USE GlaxoSmithKline LLC (US) 2012-09-12 EP disclosed
WO-2011054841-A1 TETRAHYDROQUINOLINE DERIVATIVES AND THEIR PHARMACEUTICAL USE GLAXOSMITHKLINE LLC (US) 2011-05-12 WO disclosed