SCHEMBL18791099

SCHEMBL18791099

CC1(C)OC2=C(C(=O)C(=O)c3ccccc32)C1N=[N+]=[N-]

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 6/20 0.46
IDO1 P14902 12/20 0.45
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
CES2 O00748 1/20 0.39
GMNN O75496 1/20 0.39
TDP2 O95551 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
GLA P06280 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
HSPD1 P10809 1/20 0.39
THRB P10828 1/20 0.39
CYP2C9 P11712 1/20 0.39
ALOX15 P16050 1/20 0.39
POR P16435 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18790872 0.90 IDO1 (0.56) NQO1IDO1
SCHEMBL18791135 0.82 IDO1 (0.50) NQO1IDO1KDM4EMEN1CES2
SCHEMBL103949 0.75 IDO1 (0.53) NQO1IDO1KDM4EMEN1CES2
SCHEMBL18791133 0.74 IDO1 (0.63) NQO1IDO1KDM4EMEN1CES2
SCHEMBL18791100 0.74 IDO1 (0.55) NQO1IDO1KDM4EMEN1CES2
SCHEMBL20811248 0.74 IDO1 (0.59) NQO1IDO1KDM4EMEN1CES2
SCHEMBL18791130 0.69 IDO1 (0.47) NQO1IDO1KDM4EMEN1CES2
SCHEMBL20811039 0.69 NQO1 (0.76) NQO1IDO1KDM4EMEN1CES2
SCHEMBL20811355 0.67 NQO1 (0.76) NQO1IDO1MEN1MAPTRAB9A
SCHEMBL23457125 0.65 NQO1 (0.73) NQO1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017070012-A1 LAPACHONE DERIVATIVES CONTAINING TWO REDOX CENTERS AND METHODS OF USE THEREOF THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2017-04-27 WO disclosed