SCHEMBL187916

SCHEMBL187916

[c]1ccc2[nH]c(CCN3CCCC3)cc2c1

nearest known ligand 0.67

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 9/20 0.67
CHRNA7 P36544 2/20 0.49
HRH4 Q9H3N8 1/20 0.38
MEN1 O00255 1/20 0.37
SLC6A3 Q01959 1/20 0.37
HTR2A P28223 2/20 0.36
HTR2C P28335 2/20 0.36
MBTD1 Q05BQ5 1/20 0.36
L3MBTL3 Q96JM7 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
MPO P05164 1/20 0.35
DRD2 P14416 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31061131 0.80 HRH3 (1.00) HRH3CHRNA7HRH4SLC6A3HTR2A
SCHEMBL10508496 0.79 HRH3 (0.97) HRH3CHRNA7HRH4SLC6A3HTR2A
SCHEMBL694595 0.74 ADORA1 (0.39) HRH3CHRNA7MEN1MPO
SCHEMBL5178946 0.74 MTNR1A (0.36) HRH3CHRNA7
SCHEMBL8485537 0.73 HRH3 (0.62) HRH3CHRNA7HRH4MEN1SLC6A3
SCHEMBL23482001 0.72 HRH3 (0.60) HRH3CHRNA7MEN1DRD2
SCHEMBL5778675 0.72 RHEB (0.37) HRH3
SCHEMBL188218 0.71 GAA (0.35) HRH3HTR2AHTR2C
SCHEMBL1662293 0.71 CYP1A2 (0.41)
SCHEMBL2562389 0.71 RHEB (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401281-A1 PYRIMIDOPYRIMIDOINDAZOLE DERIVATIVE MSD K.K. (JP) 2012-01-04 EP disclosed
WO-2010098367-A1 PYRIMIDOPYRIMIDOINDAZOLE DERIVATIVE BANYU PHARMACEUTICAL CO.,LTD. (JP) 2010-09-02 WO disclosed