SCHEMBL18796286

SCHEMBL18796286

Clc1ccccc1Nc1nc2ccccc2nc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.54
LCK P06239 2/20 0.52
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
TSHR P16473 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
IGF1R P08069 1/20 0.47
KDM4E B2RXH2 3/20 0.46
NPSR1 Q6W5P4 2/20 0.46
RXFP1 Q9HBX9 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
ALDH1A1 P00352 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
C1R P00736 1/20 0.45
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
KMT2A Q03164 2/20 0.44
POLB P06746 1/20 0.44
RAD52 P43351 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18795879 0.82 LCK (0.57) PDE5ALCKNPC1RAB9ATSHR
SCHEMBL14301179 0.82 PDE5A (0.51) PDE5ALCKNPC1RAB9ATSHR
SCHEMBL2243695 0.81 KDM4E (0.50) PDE5ANPC1RAB9ATSHRTDP1
SCHEMBL18323559 0.77 TDP1 (0.54) PDE5ATDP1KDM4ENPSR1RXFP1
SCHEMBL28705750 0.75 KDM4E (0.41) PDE5ANPC1RAB9ATDP1KDM4E
SCHEMBL1788978 0.74 KDM4E (0.65) KDM4ENPSR1RXFP1L3MBTL1ALDH1A1
SCHEMBL17007682 0.73 ALDH1A1 (0.51) PDE5ATSHRTDP1KDM4ENPSR1
SCHEMBL17432139 0.73 MEN1 (0.54) PDE5ALCKTDP1KDM4ENPSR1
SCHEMBL462643 0.72 TDP1 (0.58) RAB9ATDP1KDM4ENPSR1RXFP1
SCHEMBL14067142 0.72 TDP1 (0.58) TDP1KDM4ENPSR1RXFP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3368514-A1 TRISUBSTITUTEDSILYLPHENOXYHETEROCYCLES AND ANALOGUES Bayer CropScience Aktiengesellschaft (DE) 2018-09-05 EP disclosed
WO-2017072283-A1 TRISUBSTITUTEDSILYLPHENOXYHETEROCYCLES AND ANALOGUES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2017-05-04 WO disclosed