SCHEMBL18819085

SCHEMBL18819085

Cn1c(=O)n(Cc2cc(C(C)(O)C(F)(F)F)no2)c(=O)c2c1ncn2CC1CCCCC1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 15/20 0.43
KMT2A Q03164 2/20 0.42
HTT P42858 1/20 0.39
RXFP1 Q9HBX9 1/20 0.38
PARG Q86W56 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17682257 0.83 ADORA2B (0.47) KMT2ARXFP1
SCHEMBL18819720 0.82 TRPA1 (0.42) TRPA1KMT2ARXFP1
SCHEMBL18819561 0.82 KMT2A (0.41) TRPA1KMT2AHTTRXFP1
SCHEMBL20182665 0.81 TRPA1 (0.44) TRPA1KMT2AHTTRXFP1PARG
SCHEMBL19607601 0.81 KMT2A (0.44) TRPA1KMT2ARXFP1
SCHEMBL18819630 0.79 KMT2A (0.42) TRPA1KMT2ARXFP1
SCHEMBL18819717 0.78 TRPA1 (0.41) TRPA1KMT2ARXFP1
SCHEMBL17682175 0.78 KMT2A (0.42) TRPA1KMT2AHTTRXFP1
SCHEMBL24611642 0.78 MAPK1 (0.46) TRPA1KMT2AHTTRXFP1
SCHEMBL24611641 0.78 KMT2A (0.43) TRPA1KMT2ARXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017071606-A1 MEDICAL USE OF HYDROXYL PURINE COMPOUND 南京明德新药研发股份有限公司 2017-05-04 WO disclosed