SCHEMBL18824244

SCHEMBL18824244

CC(C)(C)OC(=O)NCCN1CCN(C(N)=O)CC1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 11/20 0.54
CACNA1H O95180 1/20 0.53
SIGMAR1 Q99720 3/20 0.50
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
ACKR3 P25106 1/20 0.42
CD274 Q9NZQ7 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GFER P55789 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18824235 0.95 DRD2 (0.50) DRD2CACNA1HSIGMAR1MAOAMAOB
SCHEMBL31301242 0.89 DRD2 (0.63) DRD2CACNA1HSIGMAR1TDP1CD274
SCHEMBL15859325 0.87 DRD2 (0.55) DRD2CACNA1HSIGMAR1TDP1ACKR3
SCHEMBL31496727 0.85 DRD2 (0.56) DRD2CACNA1HSIGMAR1MAOAMAOB
SCHEMBL13202614 0.84 DRD2 (0.59) DRD2CACNA1HSIGMAR1TDP1CD274
Hydrochloric Acid SCHEMBL25170707 0.84 DRD2 (0.55) DRD2CACNA1HSIGMAR1MAOAMAOB
SCHEMBL5324032 0.83 DRD2 (0.57) DRD2CACNA1HSIGMAR1TDP1CD274
SCHEMBL18390128 0.83 DRD2 (0.57) DRD2CACNA1HSIGMAR1TDP1CD274
SCHEMBL31301250 0.83 DRD2 (0.56) DRD2CACNA1HSIGMAR1TDP1CD274
SCHEMBL24172673 0.83 DRD2 (0.56) DRD2CACNA1HSIGMAR1TDP1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180312493-A1 Antibiotic Compounds, Pharmaceutical Formulations Thereof And Methods And Uses Therefor CENTRE FOR DRUG RESEARCH AND DEVELOPMENT (CA) 2018-11-01 US disclosed
WO-2017075694-A1 ANTIBIOTIC COMPOUNDS, PHARMACEUTICAL FORMULATIONS THEREOF AND METHODS AND USES THEREFOR SIMON FRASER UNIVERSITY (CA) 2017-05-11 WO disclosed
WO-2017075694-A1 ANTIBIOTIC COMPOUNDS, PHARMACEUTICAL FORMULATIONS THEREOF AND METHODS AND USES THEREFOR SIMON FRASER UNIVERSITY (CA) 2017-05-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180312493-A1 Antibiotic Compounds, Pharmaceutical Formulations Thereof And Methods And Uses Therefor UGT1A8, CYP2C8, CXCL8 DRD2 4251/4885CACNA1H 4003/4885SIGMAR1 1148/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.