SCHEMBL18828486

SCHEMBL18828486

BrC(Br)(I)COCc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.58
KDM4E B2RXH2 1/20 0.53
POLB P06746 1/20 0.53
CA1 P00915 4/20 0.43
IDO1 P14902 1/20 0.43
AGXT P21549 1/20 0.41
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CA9 Q16790 2/20 0.40
TACR1 P25103 2/20 0.39
ALDH1A1 P00352 2/20 0.38
TRPA1 O75762 1/20 0.37
NAAA Q02083 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8570364 0.82 TSHR (0.64) TSHRKDM4EPOLBCA1IDO1
SCHEMBL4788457 0.81 KDM4E (0.61) TSHRKDM4EPOLBCA1IDO1
SCHEMBL11146323 0.79 TSHR (0.67) TSHRKDM4EPOLBCA1IDO1
SCHEMBL6043011 0.78 TSHR (0.58) TSHRKDM4EPOLBCA1IDO1
SCHEMBL8570929 0.76 TSHR (0.61) TSHRKDM4EPOLBCA1IDO1
SCHEMBL1691827 0.76 TSHR (0.61) TSHRKDM4EPOLBCA1IDO1
SCHEMBL8157722 0.76 ALDH1A1 (0.61) TSHRKDM4EPOLBCA1IDO1
SCHEMBL21408338 0.76 KDM4E (0.78) TSHRKDM4EPOLBCA1IDO1
SCHEMBL5311581 0.75 TSHR (1.00) TSHRKDM4EPOLBCA1IDO1
SCHEMBL27380 0.75 TSHR (1.00) TSHRKDM4EPOLBCA1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2931708-B1 CYCLOPROPYLBORONIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF DIVERCHIM (FR) 2017-05-10 EP disclosed