SCHEMBL18833765

SCHEMBL18833765

Cc1nc2c(c(=O)[nH]c(=O)n2C)n1COCC[Si](C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
HPGD P15428 3/20 0.48
MAPK1 P28482 3/20 0.47
MAPT P10636 1/20 0.46
CYP2C9 P11712 1/20 0.45
HSD17B10 Q99714 1/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
GAA P10253 1/20 0.43
LMNA P02545 3/20 0.43
HTT P42858 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
TSHR P16473 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL638535 0.86 MAPT (0.59) ALDH1A1HPGDMAPK1MAPTHSD17B10
SCHEMBL17609629 0.84 HSD17B10 (0.47) ALDH1A1HPGDMAPK1MAPTCYP2C9
SCHEMBL16122929 0.80 MLKL (0.53) ALDH1A1MAPK1LMNAHTTSMN1; SMN2
SCHEMBL16058635 0.77 ALDH1A1 (0.41) ALDH1A1HPGDMAPK1MAPTCYP2C9
SCHEMBL16363925 0.76 MAPK1 (0.46) ALDH1A1HPGDMAPK1MAPTMEN1
SCHEMBL17609493 0.75 SMN1; SMN2 (0.55) ALDH1A1HPGDMAPK1MEN1KMT2A
SCHEMBL24476658 0.74 MAPK1 (0.69) ALDH1A1HPGDMAPK1MAPTHSD17B10
SCHEMBL9390364 0.73 HPGD (0.51) ALDH1A1HPGDMAPK1MAPTCYP2C9
SCHEMBL17609947 0.73 TRPA1 (0.47) MAPK1GAALMNAHTTSMN1; SMN2
SCHEMBL24476692 0.73 KDM4E (0.66) ALDH1A1HPGDMAPK1MAPTCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970303-B9 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES INC (US) 2017-09-20 EP disclosed
EP-2970303-B1 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES INC (US) 2017-05-10 EP disclosed