SCHEMBL1887873

SCHEMBL1887873

CC(=O)c1cn(C)c2ccccc12

nearest known ligand 0.71

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.67
POLB P06746 1/20 0.67
BRD4 O60885 1/20 0.66
L3MBTL1 Q9Y468 1/20 0.66
LMNA P02545 3/20 0.65
KMT2A Q03164 3/20 0.65
ALDH1A1 P00352 2/20 0.65
MITF O75030 1/20 0.65
MAPT P10636 1/20 0.65
NPSR1 Q6W5P4 1/20 0.65
HTT P42858 1/20 0.65
CREBBP Q92793 2/20 0.59
SMN1; SMN2 Q16637 2/20 0.58
MEN1 O00255 1/20 0.54
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
KAT2B Q92831 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29848366 1.00 NR4A2 (0.67) NR4A2POLBBRD4L3MBTL1LMNA
SCHEMBL4510662 0.87 LMNA (0.65) NR4A2POLBBRD4L3MBTL1LMNA
SCHEMBL14828742 0.85 ALDH1A1 (0.63) NR4A2POLBLMNAKMT2AALDH1A1
SCHEMBL535878 0.85 POLB (0.72) NR4A2POLBLMNAKMT2AALDH1A1
SCHEMBL29965768 0.85 POLB (0.72) NR4A2POLBLMNAKMT2AALDH1A1
Hydrochloric Acid SCHEMBL2434452 0.83 POLB (0.70) NR4A2POLBLMNAKMT2AALDH1A1
SCHEMBL30958431 0.83 LMNA (0.68) NR4A2POLBLMNAKMT2AALDH1A1
SCHEMBL2434450 0.83 LMNA (0.68) NR4A2POLBLMNAKMT2AALDH1A1
SCHEMBL2174829 0.83 NR4A2 (0.65) NR4A2POLBLMNAKMT2AALDH1A1
Indole SCHEMBL27623487 0.83 NR4A2 (0.49) NR4A2POLBBRD4L3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 417 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115974788-B Method for synthesizing alpha-straight-chain alkyl substituted heteroarene 苏州大学 2025-06-17 CN claimed
CN-106366072-B A kind of preparation method of AZD9291 上海工程技术大学 2018-12-07 CN claimed
CN-106366072-A Preparation method of AZD9291 上海工程技术大学 2017-02-01 CN claimed
EP-1778176-B1 COMPOSITION FOR COLOURING KERATIN-CONTAINING FIBRES HENKEL AG & CO KGAA (DE) 2012-07-25 EP claimed
US-7413579-B2 Method for dyeing fibers containing keratin HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2008-08-19 US claimed
EP-1432388-B1 AGENT FOR COLOURING FIBRES CONTAINING KERATIN HENKEL AG & CO KGAA (DE) 2008-06-18 EP claimed
EP-1909913-A1 METHOD FOR QUICKLY CONCEALING THE ROOTS OF HAIR THAT HAVE GROWN AFTER THE HAIR HAS BEEN DYED HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2008-04-16 EP claimed
US-7300472-B2 Agents for coloring fibers containing keratin HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2007-11-27 US claimed
EP-1789015-A1 METHOD FOR STYLISHLY CHANGING THE COLOR OF KERATINIC FIBERS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2007-05-30 EP claimed
EP-1778176-A2 MEANS FOR COLOURING KERATIN-CONTAINING FIBRES Henkel Kommanditgesellschaft auf Aktien (DE) 2007-05-02 EP claimed
EP-1432388-A1 AGENT FOR COLOURING FIBRES CONTAINING KERATIN Henkel Kommanditgesellschaft auf Aktien (DE) 2004-06-30 EP claimed
EP-1432428-A1 Agent for colouring fibres containing keratin Henkel Kommanditgesellschaft auf Aktien (DE) 2004-06-30 EP claimed
EP-1433469-A1 Composition for dyeing keratinous fibres Henkel Kommanditgesellschaft auf Aktien (DE) 2004-06-30 EP claimed
WO-2004022016-A1 AGENTS USED FOR DYEING KERATINOUS FIBERS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2004-03-18 WO claimed
WO-2003030845-A1 AGENT FOR THE COLORATION OF KERATIN-CONTAINING FIBERS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2003-04-17 WO claimed
WO-2003030847-A1 AGENT FOR COLOURING FIBRES CONTAINING KERATIN HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2003-04-17 WO claimed
WO-2003030842-A1 AGENT FOR COLOURING FIBRES CONTAINING KERATIN HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2003-04-17 WO claimed
EP-1300133-A2 Agent for dyeing keratinous fibres Henkel Kommanditgesellschaft auf Aktien (DE) 2003-04-09 EP claimed
EP-1300132-A2 Agent for dyeing keratinous fibres Henkel Kommanditgesellschaft auf Aktien (DE) 2003-04-09 EP claimed
EP-0873744-A2 Use of heterocyclic carbonyl compounds for dying keratinous fibers Henkel Kommanditgesellschaft auf Aktien (DE) 1998-10-28 EP claimed