SCHEMBL1888967

SCHEMBL1888967

CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)O.O=C(c1ncc[nH]1)c1ncc[nH]1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.59
PTPN1 P18031 3/20 0.55
CTSS P25774 3/20 0.53
CTSK P43235 2/20 0.53
CTSL P07711 1/20 0.53
CTSB P07858 1/20 0.53
ITGB3 P05106 1/20 0.51
ITGA2B P08514 1/20 0.51
PPARA Q07869 5/20 0.49
PPARG P37231 4/20 0.49
APP P05067 1/20 0.48
MAPK1 P28482 1/20 0.48
POLB P06746 1/20 0.48
MAPT P10636 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
PPARD Q03181 2/20 0.47
AKT1 P31749 1/20 0.47
ATM Q13315 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1888965 1.00 ACE (0.59) ACEPTPN1CTSSCTSKCTSL
SCHEMBL3470656 0.90 PTPN1 (0.47) ACEPTPN1CTSSCTSKCTSL
SCHEMBL1889046 0.89 CTSS (0.55) ACEPTPN1CTSSCTSKCTSL
SCHEMBL27909397 0.84 ACE (0.79) ACEPTPN1CTSSCTSKCTSL
SCHEMBL21473784 0.84 ACE (0.79) ACEPTPN1CTSSCTSKCTSL
SCHEMBL795685 0.84 ACE (0.79) ACEPTPN1CTSSCTSKCTSL
SCHEMBL66220 0.84 ACE (0.79) ACEPTPN1CTSSCTSKCTSL
SCHEMBL67020 0.84 ACE (0.79) ACEPTPN1CTSSCTSKCTSL
SCHEMBL606309 0.84 ACE (0.79) ACEPTPN1CTSSCTSKCTSL
Water SCHEMBL15362013 0.83 ACE (0.77) ACEPTPN1CTSSCTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011061675-A1 PROCESS FOR ENANTIOSELECTIVE PREPARATION OF NITROKETONE, AN INTERMEDIATE OF PROTEASE INHIBITORS PIRAMAL HEALTHCARE LIMITED (IN) 2011-05-26 WO disclosed
EP-0769003-B1 AMINO ACID-DERIVED DIAMINOPROPANOLS PHARMECO LAB INC (US) 2001-05-16 EP disclosed
EP-1059285-A2 Process for the preparation of 1,3-diamino-2-propanol and 1,3-diamino-2-propanone derivatives Pharm-Eco Laboratories, Inc. (US) 2000-12-13 EP disclosed
US-6063963-A Amino acid-derived diaminopropanols PHARM-ECO LABORATORIES, INC. (US) 2000-05-16 US disclosed
US-5631405-A Method of forming amino acid-derived diaminopropanols useful as chemical intermediates for protease-inhibitors PHARM-ECO LABORATORIES, INCORPORATED (US) 1997-05-20 US disclosed
EP-0769003-A1 AMINO ACID-DERIVED DIAMINOPROPANOLS Pharmeco Laboratories, Inc. (US) 1997-04-23 EP disclosed
US-5618966-A Method forming protease inhibitor synthetic intermediates PHARM-ECO LABORATORIES, INCORPORATED (US) 1997-04-08 US disclosed
US-5599994-A Amino acid-derived diaminopropanols PHARM-ECO LABORATORIES, INC. (US) 1997-02-04 US disclosed
WO-1996001788-A2 AMINO ACID-DERIVED DIAMINOPROPANOLS PHARM-ECO LABORATORIES, INCORPORATED (US) 1996-01-25 WO disclosed
US-5475138-A Method preparing amino acid-derived diaminopropanols PHARM-ECO LABORATORIES INCORPORATED (US) 1995-12-12 US disclosed