SCHEMBL18901372

SCHEMBL18901372

O=C(CNI)c1ccc(F)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.55
RAB9A P51151 2/20 0.55
PTPN1 P18031 1/20 0.55
PLOD2 O00469 1/20 0.53
MAPT P10636 3/20 0.49
ALDH1A1 P00352 2/20 0.49
AGTR1 P30556 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
HTR7 P34969 1/20 0.48
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
LMNA P02545 1/20 0.47
MEN1 O00255 1/20 0.47
HPGD P15428 1/20 0.47
ALOX12 P18054 1/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2491432 0.80 PLOD2 (0.69) NPC1RAB9APTPN1PLOD2MAPT
SCHEMBL13838823 0.79 NPC1 (0.61) NPC1RAB9APTPN1PLOD2MAPT
SCHEMBL2299475 0.79 NPC1 (0.55) NPC1RAB9APTPN1PLOD2MAPT
SCHEMBL1266504 0.78 NPC1 (0.64) NPC1RAB9APTPN1PLOD2MAPT
Hydrochloric Acid SCHEMBL3856160 0.78 NPC1 (0.53) NPC1RAB9APTPN1PLOD2MAPT
SCHEMBL15973607 0.78 MAPT (0.58) NPC1RAB9APTPN1PLOD2MAPT
Hydrochloric Acid SCHEMBL10472529 0.78 NPC1 (0.53) NPC1RAB9APTPN1PLOD2MAPT
SCHEMBL15020831 0.78 ALDH1A1 (0.56) NPC1RAB9APTPN1PLOD2MAPT
SCHEMBL19022048 0.77 NPC1 (0.69) NPC1RAB9APTPN1PLOD2ALDH1A1
SCHEMBL7440297 0.76 KMT2A (0.54) NPC1RAB9APTPN1PLOD2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3016951-B1 TRICYCLIC PYRIDO-CARBOXAMIDE DERIVATIVES AS ROCK INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-05-31 EP disclosed