SCHEMBL18901931

SCHEMBL18901931

COc1ccc2c(CC(=O)O)nccc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.54
AKR1C3 P42330 1/20 0.54
AKR1C2 P52895 1/20 0.54
PDE10A Q9Y233 4/20 0.52
PDE3B Q13370 2/20 0.52
PDE3A Q14432 2/20 0.52
KDM4E B2RXH2 3/20 0.47
MAPK1 P28482 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HSD17B10 Q99714 2/20 0.47
CYP1A2 P05177 2/20 0.46
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
LMNA P02545 1/20 0.46
PTGS2 P35354 2/20 0.46
LCK P06239 1/20 0.45
DYRK1A Q13627 1/20 0.45
PLAU P00749 1/20 0.44
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31207160 0.83 DYRK1A (0.57) PDE10APDE3BPDE3AKDM4EMAPK1
SCHEMBL2612055 0.80 PDE10A (0.51) PDE10APDE3BPDE3AKDM4EMAPK1
SCHEMBL30050820 0.79 PDE10A (0.50) PDE10APDE3BPDE3AKDM4EMAPK1
SCHEMBL753230 0.78 LMNA (0.52) PTGS1AKR1C3AKR1C2PDE10APDE3B
SCHEMBL13147208 0.75 TRPA1 (0.53) PTGS1AKR1C3AKR1C2PDE10APDE3B
SCHEMBL7925457 0.74 MTNR1A (0.61) PTGS1AKR1C3AKR1C2KDM4EHSD17B10
SCHEMBL31429834 0.74 MTNR1A (0.61) PTGS1AKR1C3AKR1C2KDM4EHSD17B10
SCHEMBL2540127 0.73 TRPA1 (0.50) PDE10APDE3BPDE3AKDM4EMAPK1
SCHEMBL3739311 0.73 TDP1 (0.53) KDM4ENPSR1HSD17B10LMNAPLAU
SCHEMBL11466749 0.72 PTGS1 (0.59) PTGS1AKR1C3AKR1C2KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2328865-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-05-31 EP disclosed