SCHEMBL18922705

SCHEMBL18922705

CC(S)C(=O)c1cn(-c2ccccn2)c2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 11/20 0.53
ALDH1A1 P00352 3/20 0.40
HTR7 P34969 2/20 0.40
NR4A2 P43354 1/20 0.39
MAPT P10636 2/20 0.39
HPGD P15428 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
MAPK1 P28482 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 1/20 0.39
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15440779 0.90 HTR3A (0.54) HTR3AALDH1A1HTR7NR4A2LMNA
SCHEMBL15444633 0.84 HTR3A (0.56) HTR3AALDH1A1HTR7NR4A2LMNA
SCHEMBL6044056 0.81 HTR3A (0.53) HTR3AHTR7NR4A2KDM4EPOLB
SCHEMBL15420930 0.79 NR4A2 (0.64) HTR3AALDH1A1NR4A2MAPTKDM4E
SCHEMBL20080348 0.79 KMT2A (0.52) HTR3AALDH1A1HTR7MAPTNPSR1
SCHEMBL20080410 0.78 HTR3A (0.51) HTR3AALDH1A1HTR7NR4A2MAPT
SCHEMBL19068191 0.78 HTR3A (0.54) HTR3AALDH1A1NR4A2
SCHEMBL17170671 0.76 HTR3A (0.57) HTR3AALDH1A1NR4A2LMNASMN1; SMN2
SCHEMBL17170607 0.76 ALDH1A1 (0.53) HTR3AALDH1A1NR4A2LMNASMN1; SMN2
SCHEMBL15441066 0.75 HTR3A (0.55) HTR3AALDH1A1MAPTHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9670229-B2 5-HT3 receptor antagonists TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-06-06 US disclosed