SCHEMBL18924353

SCHEMBL18924353

CCc1nc(C)c2occc2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
ADORA2A P29274 7/20 0.37
ADORA1 P30542 7/20 0.37
TSHR P16473 5/20 0.32
NPSR1 Q6W5P4 3/20 0.32
PRNP P04156 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
MAPK1 P28482 1/20 0.31
LMNA P02545 4/20 0.31
MAPT P10636 4/20 0.31
ALDH1A1 P00352 3/20 0.31
HSD17B10 Q99714 1/20 0.31
USP2 O75604 1/20 0.31
HRH4 Q9H3N8 1/20 0.31
KDM4E B2RXH2 2/20 0.31
ADORA3 P0DMS8 1/20 0.30
ADORA2B P29275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19523162 0.77 ADORA1 (0.38) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL14213484 0.76 CYP2A6 (0.33) PDE4APDE4BPDE4CPDE4DLMNA
SCHEMBL7607941 0.73 KDM4E (0.35) LMNAMAPTALDH1A1KDM4E
SCHEMBL22161609 0.73 CYP2A6 (0.31)
SCHEMBL14213485 0.73 HSD17B10 (0.50) ADORA2AMAPTALDH1A1HSD17B10
SCHEMBL21341741 0.70 ALDH1A1 (0.31) ADORA2AADORA1TSHRPRNPRXFP1
SCHEMBL20691176 0.70 ALDH1A1 (0.36) ADORA2AADORA1TSHRLMNAMAPT
SCHEMBL18211812 0.70 AURKA (0.32) ADORA2AADORA1PRNPRXFP1MAPT
SCHEMBL16840458 0.70 NUDT1 (0.39) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL14985883 0.69 GPR3 (0.55) TSHRNPSR1PRNPRXFP1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9670196-B2 Thiazole-substituted aminoheteroaryls as Spleen Tyrosine Kinase inhibitors MERCK SHARP & DOHME CORP. (US) 2017-06-06 US disclosed