SCHEMBL18924461

SCHEMBL18924461

CN(C(=O)c1ccc(-c2ccc3[nH]ccc3c2)c(F)c1)C1CCCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.47
FEN1 P39748 3/20 0.45
ALOX5AP P20292 1/20 0.45
POLB P06746 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
PDK2 Q15119 1/20 0.42
AR P10275 1/20 0.42
USP30 Q70CQ3 1/20 0.42
FASN P49327 4/20 0.41
BRD4 O60885 1/20 0.40
TAF1 P21675 1/20 0.40
CECR2 Q9BXF3 1/20 0.40
BRD9 Q9H8M2 1/20 0.40
WDR5 P61964 2/20 0.39
TRPV3 Q8NET8 1/20 0.39
GHSR Q92847 1/20 0.39
CNR2 P34972 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18924455 0.88 MAPK14 (0.43) MAPK14POLBNPC1RAB9APDK2
SCHEMBL10762514 0.85 RAB9A (0.52) POLBNPC1RAB9ABRD4CNR2
SCHEMBL18924399 0.85 MAPK14 (0.51) MAPK14POLBNPC1RAB9APDK2
SCHEMBL20897035 0.84 RAB9A (0.54) POLBNPC1RAB9ABRD4CNR2
SCHEMBL16323788 0.82 FASN (0.62) FASN
SCHEMBL18924459 0.82 FASN (0.56) MAPK14FEN1ALOX5APNPC1PDK2
SCHEMBL18924393 0.80 FASN (0.51) POLBNPC1RAB9AARFASN
SCHEMBL19391081 0.80 ABL1 (0.45) POLBNPC1RAB9AFASNBRD4
SCHEMBL18924475 0.78 FASN (0.47) FASN
SCHEMBL18924350 0.78 FASN (0.44) NPC1FASNGHSRCNR2SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9670142-B2 1,3-diaminocyclopentane carboxamide derivatives MERCK PATENT GMBH (DE) 2017-06-06 US disclosed