SCHEMBL18924561

SCHEMBL18924561

COc1ccc(-c2ccc(C(=O)N(C)C3CCCC3)cc2)c(C)c1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 4/20 0.64
MAPK14 Q16539 1/20 0.49
KMT2A Q03164 3/20 0.49
MEN1 O00255 2/20 0.49
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
POLB P06746 1/20 0.44
CNR2 P34972 1/20 0.44
OXTR P30559 2/20 0.44
AVPR1A P37288 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
S1PR1 P21453 1/20 0.42
S1PR3 Q99500 1/20 0.42
TRPM8 Q7Z2W7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18924431 0.87 MAPK14 (0.53) MCHR1MAPK14KMT2AMEN1NPC1
SCHEMBL18924429 0.85 MAPK14 (0.53) MCHR1MAPK14KMT2AMEN1NPC1
SCHEMBL18924563 0.85 MCHR1 (0.59) MCHR1KMT2AMEN1NPC1RAB9A
SCHEMBL11406234 0.82 KMT2A (0.64) MCHR1KMT2AMEN1NPC1RAB9A
SCHEMBL10454995 0.82 KMT2A (0.64) MCHR1KMT2AMEN1NPC1RAB9A
SCHEMBL16322802 0.80 FASN (0.65) MCHR1
SCHEMBL18924453 0.75 MAPK14 (0.59) MCHR1MAPK14KMT2AMEN1NPC1
SCHEMBL18924450 0.75 MAPK14 (0.58) MCHR1MAPK14KMT2AMEN1NPC1
SCHEMBL4085836 0.75 HSD17B1 (0.64) MCHR1KMT2AMEN1RAB9AMAPT
SCHEMBL3455720 0.75 SMN1; SMN2 (0.54) KMT2AMEN1NPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9670142-B2 1,3-diaminocyclopentane carboxamide derivatives MERCK PATENT GMBH (DE) 2017-06-06 US disclosed