SCHEMBL18924455

SCHEMBL18924455

Cc1cc(C(=O)N(C)C2CCCC2)ccc1-c1ccc2[nH]ccc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.43
POLB P06746 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
CNR2 P34972 1/20 0.43
AR P10275 1/20 0.43
PDK2 Q15119 1/20 0.41
PARP10 Q53GL7 1/20 0.40
PARP11 Q9NR21 1/20 0.40
BRD4 O60885 1/20 0.40
TAF1 P21675 1/20 0.40
CECR2 Q9BXF3 1/20 0.40
BRD9 Q9H8M2 1/20 0.40
LMNA P02545 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
S1PR1 P21453 1/20 0.38
MAP3K11 Q16584 2/20 0.38
ITK Q08881 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18924461 0.88 MAPK14 (0.47) MAPK14POLBNPC1RAB9ACNR2
SCHEMBL10762514 0.86 RAB9A (0.52) POLBNPC1RAB9ACNR2BRD4
SCHEMBL20897035 0.85 RAB9A (0.54) POLBNPC1RAB9ACNR2BRD4
SCHEMBL18924350 0.84 FASN (0.44) NPC1CNR2SLC6A2SLC6A4SLC6A3
SCHEMBL16323327 0.82 FASN (0.57)
SCHEMBL18924393 0.81 FASN (0.51) POLBNPC1RAB9AARMAP3K11
SCHEMBL19391081 0.81 ABL1 (0.45) POLBNPC1RAB9ABRD4SLC6A2
SCHEMBL2926458 0.79 POLB (0.55) MAPK14POLBNPC1RAB9ACNR2
SCHEMBL18924529 0.78 POLB (0.46) MAPK14POLBNPC1RAB9ACNR2
SCHEMBL21634069 0.78 SLC6A2 (0.47) POLBNPC1RAB9ACNR2PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9670142-B2 1,3-diaminocyclopentane carboxamide derivatives MERCK PATENT GMBH (DE) 2017-06-06 US disclosed