SCHEMBL18928142

SCHEMBL18928142

CCOC(=O)Cc1c(C)c2c(c(C)c1-c1cc(F)c3c(c1C)CCCO3)CN(C1CCC(C)(C)CC1)CC2

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 1/20 0.33
NR1I2 O75469 1/20 0.32
PDE4A P27815 2/20 0.32
KCNH2 Q12809 1/20 0.31
GRIN2B Q13224 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18928973 0.91 NR1I2 (0.34) NR1I2PDE4APTGDR2
SCHEMBL18928449 0.87 NR1I2 (0.33) NR1I2PDE4A
SCHEMBL18928129 0.83 NR1I2 (0.35) NR1I2PDE4AKCNH2PTGDR2
SCHEMBL18928972 0.82 NR1I2 (0.33) HTR4NR1I2PTGDR2
SCHEMBL18663914 0.81 NR1I2 (0.37) NR1I2
SCHEMBL18944148 0.80 NR1I2 (0.38) NR1I2
SCHEMBL18928273 0.80 NR1I2 (0.32) NR1I2PDE4A
SCHEMBL18920149 0.80 NR1I2 (0.49) NR1I2PDE4AKCNH2
SCHEMBL18664243 0.79 NR1I2 (0.36) NR1I2
SCHEMBL18928302 0.79 LMNA (0.40) NR1I2PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017093938-A1 TETRAHYDROISOQUINOLINE DERIVATIVES VIIV HEALTHCARE UK LIMITED (GB) 2017-06-08 WO disclosed