SCHEMBL18928449

SCHEMBL18928449

CCOC(=O)Cc1c(C)c2c(c(C)c1-c1cc(F)c3c(c1C)CCCO3)CN(C1CCC(C)(C)CC1)C(=O)C2

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.33
PDE4A P27815 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18928374 0.93 NR1I2 (0.34) NR1I2PDE4A
SCHEMBL18928319 0.91 NR1I2 (0.34) NR1I2PDE4A
SCHEMBL18928384 0.91 PDE4A (0.34) NR1I2PDE4A
SCHEMBL18928142 0.87 HTR4 (0.33) NR1I2PDE4A
SCHEMBL18928344 0.86 NR1I2 (0.35) NR1I2PDE4A
SCHEMBL18928448 0.84 NR1I2 (0.42) NR1I2PDE4A
SCHEMBL18928496 0.84 NR1I2 (0.34) NR1I2PDE4A
SCHEMBL18928421 0.84 HTR4 (0.35) PDE4A
SCHEMBL18928355 0.83 NR1I2 (0.36) NR1I2PDE4A
SCHEMBL18928331 0.83 NR1I2 (0.36) NR1I2PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017093938-A1 TETRAHYDROISOQUINOLINE DERIVATIVES VIIV HEALTHCARE UK LIMITED (GB) 2017-06-08 WO disclosed