SCHEMBL18933508

SCHEMBL18933508

CCC(=O)c1cn(-c2c(F)ccc(Cl)c2F)nn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.42
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
NOTUM Q6P988 7/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
KLKB1 P03952 1/20 0.37
ESRRA P11474 1/20 0.36
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.34
DDT P30046 1/20 0.33
LMNA P02545 1/20 0.33
RIPK1 Q13546 1/20 0.33
ACKR3 P25106 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20209713 0.88 KMT2A (0.39) KMT2ANPC1RAB9AALDH1A1KDM4E
SCHEMBL15933197 0.85 KMT2A (0.44) KMT2ANPC1RAB9AALDH1A1KDM4E
SCHEMBL14692497 0.84 NOTUM (0.52) KMT2ANPC1RAB9AALDH1A1KDM4E
SCHEMBL14706103 0.82 KMT2A (0.42) KMT2ANPC1RAB9AALDH1A1KDM4E
SCHEMBL18945325 0.80 RXRA (0.48) NOTUMKLKB1
SCHEMBL20263181 0.75 KMT2A (0.50) KMT2ANPC1RAB9AALDH1A1KDM4E
SCHEMBL20263208 0.74 GRIN2B (0.46) KMT2ANPC1RAB9ANOTUMSMN1; SMN2
SCHEMBL18944628 0.73 PTGS2 (0.47) KMT2AALDH1A1MAPTTSHR
SCHEMBL24380270 0.72 CA1 (0.52) KMT2ANPC1RAB9ASMN1; SMN2CA12
SCHEMBL18933509 0.72 P2RX7 (0.45) KMT2ARAB9AALDH1A1NOTUMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2739628-B1 NOVEL MACROCYCLES AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-06-07 EP disclosed