SCHEMBL18933773

SCHEMBL18933773

CC1(C)COB(c2ccc(N)cc2N)OC1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL615942 0.85 ALDH1A1 (0.38) CA1CA2
SCHEMBL10290477 0.80 ALDH1A1 (0.31)
SCHEMBL614874 0.80 KDM4E (0.37)
SCHEMBL2920762 0.79 CYP3A4 (0.32) CASP1
SCHEMBL613715 0.79 CYP3A4 (0.47) CA12CA1CA2CA9
SCHEMBL28919694 0.77 CASP1 (0.39) CASP1CA12CA1CA2CA9
SCHEMBL16974592 0.76 ALDH1A1 (0.39) CA1CA2
Hydrochloric Acid SCHEMBL16974558 0.75 ALDH1A1 (0.38) CA1CA2
SCHEMBL3186952 0.74 SNCA (0.40) CA12CA1CA2CA9
SCHEMBL1712145 0.72 CYP3A4 (0.37) CASP1CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2739628-B1 NOVEL MACROCYCLES AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-06-07 EP disclosed