SCHEMBL18936271

SCHEMBL18936271

C=C[C@H](Cc1ccccc1)NCC/C=C/C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 13/20 0.40
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
HTR1A P08908 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
DRD2 P14416 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
CNR1 P21554 1/20 0.36
SLC6A2 P23975 1/20 0.36
HTR2A P28223 1/20 0.36
SLC6A4 P31645 1/20 0.36
MC4R P32245 1/20 0.36
ADRA1A P35348 1/20 0.36
HRH1 P35367 1/20 0.36
OPRM1 P35372 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7789516 0.79 SIGMAR1 (0.53) SIGMAR1TSHREPHX1TAAR1
SCHEMBL19559843 0.73 SIGMAR1 (0.53) SIGMAR1CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL15375405 0.73 EPHX1 (0.44) SIGMAR1CYP1A2SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL11783856 0.71 LMNA (0.36) SIGMAR1ADRB2ADRB1HTR1AADORA3
SCHEMBL18435256 0.70 SIGMAR1 (0.46) SIGMAR1CYP1A2CYP3A4CYP2D6TSHR
Hydrochloric Acid SCHEMBL11784908 0.69 SIGMAR1 (0.35) SIGMAR1ADRB2ADRB1HTR1AADORA3
SCHEMBL9182989 0.68 MEN1 (0.59) SIGMAR1
SCHEMBL9182985 0.68 MEN1 (0.59) SIGMAR1
SCHEMBL25045960 0.67 SIGMAR1 (0.44) SIGMAR1CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL3829583 0.67 ACE (0.42) SIGMAR1CYP1A2EPHX1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017096315-A1 TRIAZOLE DAGL(α) INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 2017-06-08 WO disclosed