SCHEMBL18940429

SCHEMBL18940429

Cc1cc(C(=O)Nc2cn(Cc3cc(F)c(F)c(F)c3)cn2)cnc1CO

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TAS2R8 Q9NYW2 1/20 0.37
P2RY14 Q15391 1/20 0.37
RIPK1 Q13546 12/20 0.37
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
P2RX7 Q99572 2/20 0.36
MAP3K5 Q99683 1/20 0.34
NTRK1 P04629 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18940397 0.88 CDK5 (0.36) TAS2R8P2RY14RIPK1CDK5CDK5R1
SCHEMBL18961401 0.88 CDK5 (0.34) TAS2R8P2RY14RIPK1CDK5CDK5R1
SCHEMBL18940423 0.88 RIPK1 (0.36) TAS2R8P2RY14RIPK1CDK5CDK5R1
SCHEMBL18940377 0.86 CDK5 (0.33) TAS2R8P2RY14RIPK1CDK5CDK5R1
SCHEMBL18961335 0.85 TAS2R8 (0.35) TAS2R8P2RY14RIPK1CDK5CDK5R1
SCHEMBL18940435 0.84 TAS2R8 (0.36) TAS2R8P2RY14RIPK1CDK5CDK5R1
SCHEMBL18961381 0.83 CDK5 (0.42) TAS2R8RIPK1CDK5CDK5R1
SCHEMBL18940440 0.82 TAS2R8 (0.38) TAS2R8P2RY14RIPK1CDK5CDK5R1
SCHEMBL18940363 0.81 KDM4C (0.48) P2RY14RIPK1
SCHEMBL18961340 0.81 TAS2R8 (0.35) TAS2R8P2RY14RIPK1CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107922386-B 1, 4-disubstituted imidazole derivatives 大日本住友制药株式会社 2021-04-02 CN claimed
US-10807945-B2 1,4-disubstituted imidazole derivative SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2020-10-20 US claimed
US-20200268728-A1 DRUG TARGETING CANCER STEM CELL SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2020-08-27 US claimed
EP-3560494-A1 DRUG TARGETING CANCER STEM CELL Sumitomo Dainippon Pharma Co., Ltd. (JP) 2019-10-30 EP claimed
EP-3312170-A1 1,4-DI-SUBSTITUTED IMIDAZOLE DERIVATIVE Sumitomo Dainippon Pharma Co., Ltd. (JP) 2018-04-25 EP claimed
US-9828362-B2 1,4-disubstituted imidazole derivative SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2017-11-28 US claimed
US-20170166552-A1 1,4-DISUBSTITUTED IMIDAZOLE DERIVATIVE Sumitomo Pharma Co., Ltd. (JP) 2017-06-15 US claimed
US-11661397-B2 1,4-disubstituted imidazole derivative Sumitomo Pharma Co., Ltd. (JP) 2023-05-30 US disclosed
US-11661397-B2 1,4-disubstituted imidazole derivative Sumitomo Pharma Co., Ltd. (JP) 2023-05-30 US disclosed
US-11661397-B2 1,4-disubstituted imidazole derivative Sumitomo Pharma Co., Ltd. (JP) 2023-05-30 US disclosed
US-11434472-B2 Agent for removing undifferentiated iPS cells Sumitomo Pharma Co., Ltd. (JP) 2022-09-06 US disclosed
US-11434472-B2 Agent for removing undifferentiated iPS cells Sumitomo Pharma Co., Ltd. (JP) 2022-09-06 US disclosed
US-20210171440-A1 1,4-DISUBSTITUTED IMIDAZOLE DERIVATIVE Sumitomo Pharma Co., Ltd. (JP) 2021-06-10 US disclosed
EP-3312170-A1 1,4-DI-SUBSTITUTED IMIDAZOLE DERIVATIVE Sumitomo Dainippon Pharma Co., Ltd. (JP) 2018-04-25 EP disclosed
US-9828362-B2 1,4-disubstituted imidazole derivative SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2017-11-28 US disclosed
US-9828362-B2 1,4-disubstituted imidazole derivative SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2017-11-28 US disclosed
US-9828362-B2 1,4-disubstituted imidazole derivative SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2017-11-28 US disclosed
US-20170166552-A1 1,4-DISUBSTITUTED IMIDAZOLE DERIVATIVE Sumitomo Pharma Co., Ltd. (JP) 2017-06-15 US disclosed
US-20170166552-A1 1,4-DISUBSTITUTED IMIDAZOLE DERIVATIVE Sumitomo Pharma Co., Ltd. (JP) 2017-06-15 US disclosed
US-20170166552-A1 1,4-DISUBSTITUTED IMIDAZOLE DERIVATIVE Sumitomo Pharma Co., Ltd. (JP) 2017-06-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170166552-A1 1,4-DISUBSTITUTED IMIDAZOLE DERIVATIVE NR4A3, NR0B1, NR2C2 TAS2R8 1436/4885P2RY14 3931/4885RIPK1 3318/4885
US-11434472-B2 Agent for removing undifferentiated iPS cells SALL4, NR4A2, NES TAS2R8 2868/4885P2RY14 2413/4885RIPK1 3612/4885
US-20210171440-A1 1,4-DISUBSTITUTED IMIDAZOLE DERIVATIVE NR4A3, NR0B1, NR2C2 TAS2R8 1436/4885P2RY14 3931/4885RIPK1 3318/4885
US-11661397-B2 1,4-disubstituted imidazole derivative NR4A3, NR0B1, NR2C2 TAS2R8 1436/4885P2RY14 3931/4885RIPK1 3318/4885
US-20200268728-A1 DRUG TARGETING CANCER STEM CELL NR5A1, NR3C1, NR3C2 TAS2R8 2778/4885P2RY14 3207/4885RIPK1 2464/4885
US-10807945-B2 1,4-disubstituted imidazole derivative NR0B1, NR4A3, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 TAS2R8 1920/4885P2RY14 3845/4885RIPK1 2366/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.