SCHEMBL18953580

SCHEMBL18953580

COc1cc(Cl)c(Cl)c2c1NC(=O)NS2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 2/20 0.35
MAPT P10636 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HSP90AA1 P07900 1/20 0.33
PKM P14618 1/20 0.33
MAPK1 P28482 1/20 0.33
RAB9A P51151 1/20 0.33
CCR6 P51684 1/20 0.33
CACNA1B Q00975 1/20 0.33
APBA1 Q02410 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
APOBEC3G Q9HC16 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
HTR1A P08908 1/20 0.33
HTR1D P28221 1/20 0.33
HTR2C P28335 1/20 0.33
HTR7 P34969 1/20 0.33
HTR5A P47898 1/20 0.33
AKR1B1 P15121 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18953512 0.86 HTR1A (0.41) PDE7AMAPTALDH1A1HSP90AA1PKM
SCHEMBL18953701 0.79 PDE7A (0.45) PDE7AMAPTALDH1A1HSP90AA1MAPK1
SCHEMBL4686117 0.73 SERPINH1 (0.35) PDE7AMAPTALDH1A1HSP90AA1MAPK1
SCHEMBL18953654 0.73 AKR1B1 (0.36) PDE7AALDH1A1AKR1B1GRIN2DGRIN3B
SCHEMBL18953588 0.67
SCHEMBL18953486 0.67 CREBBP (0.33) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL18953378 0.67 IGF1R (0.37) PDE3BPDE3AGRIN2DGRIN3BGRIN1
SCHEMBL10571070 0.66 CRHBP (0.35) PDE7AMAPTALDH1A1HSP90AA1PKM
SCHEMBL18953531 0.64 ALDH1A1 (0.38) PDE7AALDH1A1HTR1AHTR1DHTR2C
SCHEMBL18953724 0.62 CREBBP (0.39) PDE7AALDH1A1HTR1AHTR1DHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017098421-A1 BENZOTHIADIAZINE COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-06-15 WO disclosed