SCHEMBL18955178

SCHEMBL18955178

CS(=O)(=O)c1ccccc1-c1ccc(N2CCCC(NC(=O)Nc3ccc(C(F)(F)F)cc3)C2=O)c(F)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 17/20 1.00
FPR1 P21462 7/20 0.85
F10 P00742 3/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30337884 1.00 FPR2 (1.00) FPR2FPR1F10
SCHEMBL18955163 0.92 FPR2 (1.00) FPR2FPR1F10
SCHEMBL30337813 0.92 FPR2 (1.00) FPR2FPR1F10
SCHEMBL30337635 0.91 FPR2 (0.89) FPR2FPR1F10
SCHEMBL18955189 0.91 FPR2 (0.89) FPR2FPR1F10
SCHEMBL18955269 0.91 FPR2 (0.89) FPR2FPR1F10
SCHEMBL30337618 0.91 FPR2 (0.89) FPR2FPR1F10
SCHEMBL30337558 0.91 FPR2 (0.88) FPR2FPR1F10
SCHEMBL18964535 0.91 FPR2 (0.88) FPR2FPR1F10
SCHEMBL18964046 0.91 FPR2 (0.88) FPR2FPR1F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11530183-B2 Piperidinone formyl peptide 2 receptor and formyl peptide 1 receptor agonists BRISTOL-MYERS SQUIBB COMPANY (US) 2022-12-20 US disclosed
US-11530183-B2 Piperidinone formyl peptide 2 receptor and formyl peptide 1 receptor agonists BRISTOL-MYERS SQUIBB COMPANY (US) 2022-12-20 US disclosed
US-11186544-B2 Piperidinone formyl peptide 2 receptor and formyl peptide 1 receptor agonists BRISTOL-MYERS SQUIBB COMPANY (US) 2021-11-30 US disclosed
US-11186544-B2 Piperidinone formyl peptide 2 receptor and formyl peptide 1 receptor agonists BRISTOL-MYERS SQUIBB COMPANY (US) 2021-11-30 US disclosed
EP-3414227-B1 PIPERIDINONE FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS BRISTOL MYERS SQUIBB CO (US) 2021-11-24 EP disclosed
EP-3414227-B1 PIPERIDINONE FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS BRISTOL MYERS SQUIBB CO (US) 2021-11-24 EP disclosed
US-20200299237-A1 PIPERIDINONE FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS BRISTOL MYERS SQUIBB CO (US) 2020-09-24 US disclosed
US-20200299237-A1 PIPERIDINONE FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS BRISTOL MYERS SQUIBB CO (US) 2020-09-24 US disclosed
US-10717708-B2 Piperidinone formyl peptide 2 receptor and formyl peptide 1 receptor agonists BRISTOL-MYERS SQUIBB COMPANY (US) 2020-07-21 US disclosed
US-10717708-B2 Piperidinone formyl peptide 2 receptor and formyl peptide 1 receptor agonists BRISTOL-MYERS SQUIBB COMPANY (US) 2020-07-21 US disclosed
US-20200123108-A1 PIPERIDINONE FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS BRISTOL MYERS SQUIBB CO (US) 2020-04-23 US disclosed
US-20200123108-A1 PIPERIDINONE FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS BRISTOL MYERS SQUIBB CO (US) 2020-04-23 US disclosed
EP-3634412-A1 PIPERIDINONE FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS Bristol-Myers Squibb Company (US) 2020-04-15 EP disclosed
EP-3414227-A1 PIPERIDINONE FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS Bristol-Myers Squibb Company (US) 2018-12-19 EP disclosed
WO-2018227065-A1 PIPERIDINONE FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-12-13 WO disclosed
US-20180327358-A1 PIPERIDINONE FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS SYNGENE INTERNATIONAL LIMITED (IN) 2018-11-15 US disclosed
WO-2017100390-A1 PIPERIDINONE FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2017-06-15 WO disclosed
WO-2017100390-A1 PIPERIDINONE FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2017-06-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10717708-B2 Piperidinone formyl peptide 2 receptor and formyl peptide 1 receptor agonists FPR1, FPR2, FPR3 FPR2 2/4885FPR1 1/4885F10 2404/4885
US-11186544-B2 Piperidinone formyl peptide 2 receptor and formyl peptide 1 receptor agonists FPR1, FPR2, FPR3 FPR2 2/4885FPR1 1/4885F10 2461/4885
US-20200123108-A1 PIPERIDINONE FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS FPR1, FPR2, FPR3 FPR2 2/4885FPR1 1/4885F10 2461/4885
US-20180327358-A1 PIPERIDINONE FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS FPR1, FPR2, FPR3 FPR2 2/4885FPR1 1/4885F10 2404/4885
US-11530183-B2 Piperidinone formyl peptide 2 receptor and formyl peptide 1 receptor agonists FPR1, FPR2, FPR3 FPR2 2/4885FPR1 1/4885F10 2404/4885
US-20200299237-A1 PIPERIDINONE FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS FPR1, FPR2, FPR3 FPR2 2/4885FPR1 1/4885F10 2404/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.