SCHEMBL18977640

SCHEMBL18977640

Nc1nc(C2CCCC(F)(F)CC2)no1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.35
CASP3 P42574 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NR1I2 O75469 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
NR1H4 Q96RI1 1/20 0.31
FABP4 P15090 4/20 0.31
FABP5 Q01469 4/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18978014 0.84 S1PR4 (0.33) NR1I2CYP2C9CYP2C19NR1H4
SCHEMBL18977643 0.79 POLB (0.50) POLBCASP3SENP7SENP6NPC1
SCHEMBL18977638 0.76 CHRNA7 (0.36)
SCHEMBL16364714 0.73 MAP4K4 (0.37) POLBCASP3SENP7SENP6NPC1
SCHEMBL15479741 0.71 HCRTR1 (0.37) POLBCASP3SENP7SENP6NR1I2
SCHEMBL17960915 0.69 CHRM3 (0.34)
SCHEMBL23439154 0.67 HCRTR1 (0.36) POLBCASP3SENP7SENP6NR1H4
SCHEMBL18977432 0.67 ALDH1A1 (0.36) NPC1RAB9ANR1H4
SCHEMBL16364885 0.65 MAP4K4 (0.33) NR1H4
SCHEMBL15479717 0.62 HCRTR1 (0.38) NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2703392-B1 5-MEMBERED RING AROMATIC HETEROCYCLIC DERIVATIVE HAVING NPY Y5 RECEPTOR ANTAGONISTIC ACTIVITY SHIONOGI & CO (JP) 2017-06-14 EP disclosed