SCHEMBL18978014

SCHEMBL18978014

Nc1nc(C2CCC(F)(F)C2)no1

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
S1PR4 O95977 5/20 0.33
S1PR1 P21453 5/20 0.33
S1PR3 Q99500 5/20 0.33
S1PR5 Q9H228 5/20 0.33
NR1H4 Q96RI1 4/20 0.33
CHRNA7 P36544 1/20 0.31
MAP3K12 Q12852 1/20 0.30
NR1I2 O75469 2/20 0.30
CYP2C9 P11712 2/20 0.30
CYP2C19 P33261 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18977638 0.86 CHRNA7 (0.36) CHRNA7
SCHEMBL18977640 0.84 POLB (0.35) NR1H4NR1I2CYP2C9CYP2C19
SCHEMBL16364885 0.80 MAP4K4 (0.33) S1PR4S1PR1S1PR3S1PR5NR1H4
SCHEMBL15479717 0.78 HCRTR1 (0.38) S1PR4S1PR1S1PR3S1PR5NR1H4
SCHEMBL18977643 0.71 POLB (0.50) S1PR1CYP2C9CYP2C19
SCHEMBL16364714 0.69 MAP4K4 (0.37) NR1H4NR1I2CYP2C9CYP2C19
SCHEMBL23439154 0.69 HCRTR1 (0.36) NR1H4
SCHEMBL15479741 0.67 HCRTR1 (0.37) NR1H4NR1I2CYP2C9CYP2C19
SCHEMBL18977432 0.66 ALDH1A1 (0.36) NR1H4
SCHEMBL16364833 0.65 MIF (0.36) CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2703392-B1 5-MEMBERED RING AROMATIC HETEROCYCLIC DERIVATIVE HAVING NPY Y5 RECEPTOR ANTAGONISTIC ACTIVITY SHIONOGI & CO (JP) 2017-06-14 EP disclosed