SCHEMBL18977652

SCHEMBL18977652

Nc1nc(CC2CCCCC2)no1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
RECQL P46063 1/20 0.42
HRH4 Q9H3N8 1/20 0.40
RAB9A P51151 2/20 0.40
ALDH1A1 P00352 2/20 0.40
OPRL1 P41146 1/20 0.36
NPC1 O15118 1/20 0.36
KDM4E B2RXH2 2/20 0.36
BMP1 P13497 1/20 0.35
HSD11B1 P28845 1/20 0.35
FBP1 P09467 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
GAA P10253 1/20 0.34
LMNA P02545 1/20 0.34
PDE8B O95263 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18977435 0.90 ALDH1A1 (0.41) RAB9AALDH1A1NPC1KDM4EHSD11B1
SCHEMBL18977432 0.80 ALDH1A1 (0.36) RAB9AALDH1A1NPC1KDM4EHSD11B1
SCHEMBL2655815 0.78 OPRL1 (0.41) TSHRRECQLHRH4RAB9AALDH1A1
SCHEMBL16364797 0.76 OPRL1 (0.39) TSHRRECQLHRH4RAB9AALDH1A1
SCHEMBL15479746 0.74 BMP1 (0.40) TSHRRECQLRAB9AALDH1A1OPRL1
SCHEMBL7176775 0.72 HRH4 (0.59) HRH4MEN1KMT2A
SCHEMBL16364796 0.72 KDM4E (0.38) RAB9AALDH1A1OPRL1KDM4EHSD11B1
SCHEMBL15479751 0.71 BMP1 (0.39) TSHRRECQLRAB9AALDH1A1OPRL1
SCHEMBL29161733 0.71 BMP1 (0.34) TSHRRECQLHRH4RAB9AALDH1A1
SCHEMBL29161719 0.70 SIGMAR1 (0.36) TSHRRECQLHRH4RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2703392-B1 5-MEMBERED RING AROMATIC HETEROCYCLIC DERIVATIVE HAVING NPY Y5 RECEPTOR ANTAGONISTIC ACTIVITY SHIONOGI & CO (JP) 2017-06-14 EP disclosed