Predicted protein targets (top 14)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | PDE4A | P27815 | 1/20 | 0.53 |
| ▸ | USP2 | O75604 | 1/20 | 0.50 |
| ▸ | SLCO1B1 | Q9Y6L6 | 1/20 | 0.50 |
| ▸ | LMNA | P02545 | 2/20 | 0.46 |
| ▸ | L3MBTL1 | Q9Y468 | 1/20 | 0.37 |
| ▸ | TDP1 | Q9NUW8 | 1/20 | 0.35 |
| ▸ | SLC1A1 | P43005 | 3/20 | 0.35 |
| ▸ | GRIK1 | P39086 | 1/20 | 0.33 |
| ▸ | SLC7A5 | Q01650 | 1/20 | 0.33 |
| ▸ | KDM4E | B2RXH2 | 2/20 | 0.32 |
| ▸ | PTGS1 | P23219 | 1/20 | 0.31 |
| ▸ | SLC7A11 | Q9UPY5 | 1/20 | 0.31 |
| ▸ | SLC1A3 | P43003 | 2/20 | 0.31 |
| ▸ | SLC1A2 | P43004 | 2/20 | 0.31 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL27516225 | 0.86 | PDE4A (0.58) | PDE4AUSP2SLCO1B1LMNAL3MBTL1 | |
| SCHEMBL4422883 | 0.86 | PDE4A (0.58) | PDE4AUSP2SLCO1B1LMNAL3MBTL1 | |
| SCHEMBL321750 | 0.86 | PDE4A (0.58) | PDE4AUSP2SLCO1B1LMNAL3MBTL1 | |
| SCHEMBL92769 | 0.86 | PDE4A (0.58) | PDE4AUSP2SLCO1B1LMNAL3MBTL1 | |
| Hydrochloric Acid SCHEMBL27659069 | 0.84 | PDE4A (0.56) | PDE4AUSP2SLCO1B1LMNAL3MBTL1 | |
| Bromide SCHEMBL27760150 | 0.84 | PDE4A (0.56) | PDE4AUSP2SLCO1B1LMNAL3MBTL1 | |
| Ammonia Solution, Strong SCHEMBL27782446 | 0.84 | PDE4A (0.56) | PDE4AUSP2SLCO1B1LMNAL3MBTL1 | |
| Methane SCHEMBL28111172 | 0.84 | PDE4A (0.56) | PDE4AUSP2SLCO1B1LMNAL3MBTL1 | |
| SCHEMBL6514261 | 0.80 | PDE4A (0.48) | PDE4AUSP2SLCO1B1LMNAL3MBTL1 | |
| Xylitol SCHEMBL17797759 | 0.80 | USP2 (0.61) | PDE4AUSP2SLCO1B1LMNAL3MBTL1 |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| EP-3661543-A1 | MODIFIED DDAH POLYPEPTIDES COMPRISING A PHARMACOKINETIC ENHANCING MOIETY, IMPROVED PHARMACOLOGY AND THEIR USES | Vasculonics LLC (US) | 2020-06-10 | — | — | EP | disclosed |
| WO-2020082057-A1 | INTERLEUKIN-10 POLYPEPTIDE CONJUGATES, DIMERS THEREOF, AND THEIR USES | AMBRX, INC. (US) | 2020-04-23 | — | — | WO | disclosed |
| WO-2019028040-A1 | MODIFIED DDAH POLYPEPTIDES COMPRISING A PHARMACOKINETIC ENHANCING MOIETY, IMPROVED PHARMACOLOGY AND THEIR USES | VASCULONICS LLC (US) | 2019-02-07 | — | — | WO | disclosed |
| EP-2615108-B1 | Modified human plasma polypeptide or fc scaffolds and thier uses | AMBRX INC (US) | 2016-10-26 | — | — | EP | disclosed |
| EP-2820034-A1 | MODIFIED ADIPONECTIN POLYPEPTIDES AND THEIR USES | Ambrx, Inc. (US) | 2015-01-07 | — | — | EP | disclosed |
| EP-2820033-A1 | INTERLEUKIN-10 POLYPEPTIDE CONJUGATES AND THEIR USES | Ambrx, Inc. (US) | 2015-01-07 | — | — | EP | disclosed |
| WO-2013130913-A1 | INTERLEUKIN-10 POLYPEPTIDE CONJUGATES AND THEIR USES | AMBRX, INC. (US) | 2013-09-06 | — | — | WO | disclosed |
| WO-2013130676-A1 | MODIFIED ADIPONECTIN POLYPEPTIDES AND THEIR USES | AMBRX, INC. (US) | 2013-09-06 | — | — | WO | disclosed |
| WO-2011079293-A1 | TUMOR NECROSIS FACTOR-RELATED APOPTOSIS INDUCING LIGAND POLYPEPTIDES AND THEIR USES | AMBRX, INC (US) | 2011-06-30 | — | — | WO | disclosed |
| EP-2318029-A2 | MODIFIED BOVINE G-CSF POLYPEPTIDES AND THEIR USES | Ambrx, Inc. (US) | 2011-05-11 | — | — | EP | disclosed |
| EP-1718339-A4 | MODIFIED HUMAN INTERFERON POLYPEPTIDES AND THEIR USES | AMBRX INC (US) | 2008-08-13 | — | — | EP | disclosed |
| WO-2008030558-A2 | MODIFIED HUMAN PLASMA POLYPEPTIDE OR FC SCAFFOLDS AND THEIR USES | AMBRX, INC. (US) | 2008-03-13 | — | — | WO | disclosed |
| EP-1893229-A2 | IMPROVED HUMAN INTERFERON MOLECULES AND THEIR USES | Ambrx, Inc. (US) | 2008-03-05 | — | — | EP | disclosed |
| EP-1836314-A2 | MODIFIED HUMAN GROWTH HORMONE | Ambrx, Inc. (US) | 2007-09-26 | — | — | EP | disclosed |
| WO-2006069220-A9 | MODIFIED HUMAN GROWTH HORMONE | AMBRX INC (US) | 2007-08-02 | — | — | WO | disclosed |
| WO-2006133088-A2 | IMPROVED HUMAN INTERFERON MOLECULES AND THEIR USES | AMBRX, INC. (US) | 2006-12-14 | — | — | WO | disclosed |
| WO-2006133089-A2 | IMPROVED HUMAN INTERFERON MOLECULES AND THEIR USES | AMBRX, INC. (US) | 2006-12-14 | — | — | WO | disclosed |
| EP-1718339-A2 | MODIFIED HUMAN INTERFERON POLYPEPTIDES AND THEIR USES | Ambrx, Inc. (US) | 2006-11-08 | — | — | EP | disclosed |
| WO-2006069220-A2 | MODIFIED HUMAN GROWTH HORMONE | AMBRX, INC. (US) | 2006-06-29 | — | — | WO | disclosed |
| WO-2005074524-A2 | MODIFIED HUMAN INTERFERON POLYPEPTIDES AND THEIR USES | AMBRX, INC. (US) | 2005-08-18 | — | — | WO | disclosed |