SCHEMBL18985355

SCHEMBL18985355

CCCOc1ccc(NC(=O)/C=C/c2ccc(-c3ccccc3CC)s2)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 2/20 0.47
PNLIP P16233 1/20 0.42
HDAC3 O15379 1/20 0.41
ABL1 P00519 1/20 0.41
EGFR P00533 1/20 0.41
ERBB2 P04626 1/20 0.41
INSR P06213 1/20 0.41
PDGFRB P09619 1/20 0.41
CDK2 P24941 1/20 0.41
PLK1 P53350 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18985281 0.88 NAMPT (0.49) NAMPTPNLIPHDAC3ABL1EGFR
SCHEMBL19003361 0.78 NAMPT (0.52) NAMPTPNLIPHDAC3HDAC4HDAC1
SCHEMBL18985314 0.76 MAPT (0.56) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL19003279 0.74 ALDH1A1 (0.47) NAMPTHDAC3EGFRHDAC4HDAC1
SCHEMBL19003461 0.72 EGFR (0.54) NAMPTEGFRHDAC8ALDH1A1MAPT
SCHEMBL19003312 0.72 MEN1 (0.47) NAMPTEGFRHDAC8ALDH1A1MAPT
SCHEMBL19003456 0.70 MAPT (0.48) EGFRALDH1A1HTTMAPTTP53
SCHEMBL11812683 0.68 MAPT (0.76) PNLIPEGFRERBB2ALDH1A1HTT
SCHEMBL4007931 0.67 BCHE (0.55) NAMPTEGFRBCHEACHE
SCHEMBL5108944 0.67 BCHE (0.55) NAMPTEGFRBCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102014-A1 PROPENAMIDE THIOPHENE DERIVATIVES AS FLAVIVIRUS INHIBITORS AND THEIR USE UNIVERSITE D'AIX-MARSEILLE (FR) 2017-06-22 WO claimed