SCHEMBL19002080

SCHEMBL19002080

COc1cc(N)c(C2NC(C)(C)CO2)cc1OC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 5/20 0.37
CYP3A4 P08684 2/20 0.35
MAOA P21397 3/20 0.33
TSHR P16473 2/20 0.33
HSD17B10 Q99714 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KDM4E B2RXH2 3/20 0.32
NPC1 O15118 1/20 0.32
CHRNA1 P02708 2/20 0.32
CHRNG P07510 2/20 0.32
CHRNB1 P11230 2/20 0.32
CHRNB2 P17787 2/20 0.32
CHRNB4 P30926 2/20 0.32
CHRNA3 P32297 2/20 0.32
CHRNA4 P43681 2/20 0.32
CHRND Q07001 2/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A3 Q01959 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16381560 0.75 DRD2 (0.46) MEN1KMT2AALDH1A1KDM4ESMN1; SMN2
SCHEMBL7792229 0.75 CYP2C19 (0.45) ALDH1A1TDP1KDM4ECHRNA1CHRNG
SCHEMBL10637412 0.69 CHRNA1 (0.33) KMT2AALDH1A1CHRNA1CHRNGCHRNB1
SCHEMBL7795756 0.67 CHRNA1 (0.46) ALDH1A1CYP3A4TSHRKDM4ECHRNA1
SCHEMBL4856372 0.67 CYP3A4 (0.38) MEN1KMT2AALDH1A1CYP3A4MAOA
SCHEMBL7796227 0.66 CHRNA1 (0.40) MEN1KMT2AALDH1A1NPC1CHRNA1
SCHEMBL6302031 0.66 CHRNA1 (0.50) MEN1KMT2AKDM4ENPC1CHRNA1
SCHEMBL21156708 0.65 HTR2A (0.53) CYP3A4KDM4ENPC1
SCHEMBL209984 0.63 NPC1 (0.56) MEN1KMT2AALDH1A1CYP3A4TSHR
SCHEMBL29532421 0.63 NPC1 (0.56) MEN1KMT2AALDH1A1CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017103615-A1 COMBINATION PRODUCT LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2017-06-22 WO disclosed