SCHEMBL19003464

SCHEMBL19003464

O=C(/C=C/c1ccc(Br)s1)Nc1ccc(Cl)c(Cl)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.53
MAPT P10636 9/20 0.52
TP53 P04637 4/20 0.52
CA2 P00918 1/20 0.47
CA4 P22748 1/20 0.47
CA5A P35218 1/20 0.47
CA9 Q16790 1/20 0.47
EPHX1 P07099 2/20 0.46
EPHX2 P34913 2/20 0.46
SMN1; SMN2 Q16637 3/20 0.44
THRB P10828 2/20 0.44
DHODH Q02127 1/20 0.44
KDM4E B2RXH2 3/20 0.43
TDP1 Q9NUW8 2/20 0.43
POLB P06746 1/20 0.43
MEN1 O00255 7/20 0.43
KMT2A Q03164 7/20 0.43
LMNA P02545 4/20 0.43
NPC1 O15118 4/20 0.43
HTT P42858 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19003254 0.89 EGFR (0.53) EGFRMAPTTP53SMN1; SMN2TDP1
SCHEMBL19003251 0.83 EGFR (0.68) EGFRMAPTTP53SMN1; SMN2KDM4E
SCHEMBL19003284 0.82 MAPT (0.58) MAPTTP53SMN1; SMN2POLBMEN1
SCHEMBL19003280 0.81 MAPT (0.52) MAPTTP53CA2CA4CA5A
SCHEMBL19003279 0.80 ALDH1A1 (0.47) EGFRMAPTTP53SMN1; SMN2KDM4E
SCHEMBL19003456 0.80 MAPT (0.48) EGFRMAPTTP53SMN1; SMN2THRB
SCHEMBL18985272 0.80 MAOB (0.63) EGFRMAPTTP53SMN1; SMN2MEN1
SCHEMBL19003250 0.80 MAPT (0.51) EGFRMAPTTP53SMN1; SMN2THRB
SCHEMBL19003247 0.79 MAPT (0.60) EGFRMAPTSMN1; SMN2KDM4EPOLB
SCHEMBL15708821 0.78 EPHX1 (0.68) MAPTTP53CA2CA4CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102014-A1 PROPENAMIDE THIOPHENE DERIVATIVES AS FLAVIVIRUS INHIBITORS AND THEIR USE UNIVERSITE D'AIX-MARSEILLE (FR) 2017-06-22 WO disclosed